3D-QSAR-assisted drug design: identification of a potent quinazoline-based Aurora kinase inhibitor.
about
Computational methods in drug discoveryProfiling the interaction mechanism of quinoline/quinazoline derivatives as MCHR1 antagonists: an in silico method.Discovery of BPR1K871, a quinazoline based, multi-kinase inhibitor for the treatment of AML and solid tumors: Rational design, synthesis, in vitro and in vivo evaluationFacile identification of dual FLT3-Aurora A inhibitors: a computer-guided drug design approach.Discovery of 7-aryl-substituted (1,5-naphthyridin-4-yl)ureas as aurora kinase inhibitors.Synthesis, antitumor evaluation and docking study of novel 4-anilinoquinazoline derivatives as potential epidermal growth factor receptor (EGFR) inhibitors.Novel Quinazoline Derivatives Bearing Various 4-Aniline Moieties as Potent EGFR Inhibitors with Enhanced Activity Against NSCLC Cell Lines.
P2860
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P2860
3D-QSAR-assisted drug design: identification of a potent quinazoline-based Aurora kinase inhibitor.
description
2012 nî lūn-bûn
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2012年の論文
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2012年学术文章
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name
3D-QSAR-assisted drug design: ...... based Aurora kinase inhibitor.
@en
3D-QSAR-assisted drug design: ...... based Aurora kinase inhibitor.
@nl
type
label
3D-QSAR-assisted drug design: ...... based Aurora kinase inhibitor.
@en
3D-QSAR-assisted drug design: ...... based Aurora kinase inhibitor.
@nl
prefLabel
3D-QSAR-assisted drug design: ...... based Aurora kinase inhibitor.
@en
3D-QSAR-assisted drug design: ...... based Aurora kinase inhibitor.
@nl
P2093
P2860
P50
P356
P1433
P1476
3D-QSAR-assisted drug design: ...... based Aurora kinase inhibitor.
@en
P2093
Chang-Ying Chu
Cheng-Wei Lin
Chun-Hwa Chen
Chun-Wei Chang
Hui-Yi Shiao
John T A Hsu
Teng-Kuang Yeh
Wen-Chieh Wang
Yen-Chun Lee
P2860
P304
P356
10.1002/CMDC.201200464
P577
2012-11-22T00:00:00Z