Truncation and optimisation of peptide inhibitors of cyclin-dependent kinase 2-cyclin a through structure-guided design
about
Targeting cyclin-dependent kinases in human cancers: from small molecules to Peptide inhibitorsDiscovery of a Potential Allosteric Ligand Binding Site in CDK2Iterative conversion of cyclin binding groove peptides into druglike CDK inhibitors with antitumor activityOptimization of non-ATP competitive CDK/cyclin groove inhibitors through REPLACE-mediated fragment assembly.Fragment based discovery of arginine isosteres through REPLACE: towards non-ATP competitive CDK inhibitors.Selective inhibition of proteins regulating CDK/cyclin complexes: strategy against cancer--a review.Benzamide capped peptidomimetics as non-ATP competitive inhibitors of CDK2 using the REPLACE strategy.Structural and functional analysis of cyclin D1 reveals p27 and substrate inhibitor binding requirements.
P2860
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P2860
Truncation and optimisation of peptide inhibitors of cyclin-dependent kinase 2-cyclin a through structure-guided design
description
2009 nî lūn-bûn
@nan
2009 թուականի Յուլիսին հրատարակուած գիտական յօդուած
@hyw
2009 թվականի հուլիսին հրատարակված գիտական հոդված
@hy
2009年の論文
@ja
2009年論文
@yue
2009年論文
@zh-hant
2009年論文
@zh-hk
2009年論文
@zh-mo
2009年論文
@zh-tw
2009年论文
@wuu
name
Truncation and optimisation of ...... hrough structure-guided design
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Truncation and optimisation of ...... hrough structure-guided design
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Truncation and optimisation of ...... hrough structure-guided design
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Truncation and optimisation of ...... hrough structure-guided design
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Truncation and optimisation of ...... hrough structure-guided design
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Truncation and optimisation of ...... hrough structure-guided design
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Truncation and optimisation of ...... hrough structure-guided design
@ast
Truncation and optimisation of ...... hrough structure-guided design
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Truncation and optimisation of ...... hrough structure-guided design
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P2093
P356
P1433
P1476
Truncation and optimisation of ...... hrough structure-guided design
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P2093
Andy Plater
Angela Cowan
Campbell McInnes
George Kontopidis
Lorraine Innes
Martin J Andrews
Peter M Fischer
Scott Renachowski
P2860
P304
P356
10.1002/CMDC.200900093
P577
2009-07-01T00:00:00Z