Dithiocarbamates: a new class of carbonic anhydrase inhibitors. Crystallographic and kinetic investigations
about
Dithiocarbamates Strongly Inhibit Carbonic Anhydrases and Show Antiglaucoma Action in VivoProbing the surface of human carbonic anhydrase for clues towards the design of isoform specific inhibitorsA class of 4-sulfamoylphenyl-ω-aminoalkyl ethers with effective carbonic anhydrase inhibitory action and antiglaucoma effects.Identification of metal dithiocarbamates as a novel class of antileishmanial agentsInsights towards sulfonamide drug specificity in α-carbonic anhydrasesStructure-based drug discovery of carbonic anhydrase inhibitors.Exploiting the hydrophobic and hydrophilic binding sites for designing carbonic anhydrase inhibitors.Antiglaucoma carbonic anhydrase inhibitors: a patent review.Recent advances in the discovery of zinc-binding motifs for the development of carbonic anhydrase inhibitors.Targeting tumour hypoxia to prevent cancer metastasis. From biology, biosensing and technology to drug development: the METOXIA consortium.Bacterial, fungal and protozoan carbonic anhydrases as drug targets.How many carbonic anhydrase inhibition mechanisms exist?Design, synthesis and pharmacological analysis of 5-[4'-(substituted-methyl)[1,1'-biphenyl]-2-yl]-1H-tetrazoles.Inhibition of carbonic anhydrase from Trypanosoma cruzi for the management of Chagas disease: an underexplored therapeutic opportunity.Synthesis and antitumor activity of tetrahydrocarbazole hybridized with dithioate derivatives.Advances in structure-based drug discovery of carbonic anhydrase inhibitors.Inhibition of the β-carbonic anhydrase from the dandruff-producing fungus Malassezia globosa with monothiocarbamates.Hydroxylamine-O-sulfonamide is a versatile lead compound for the development of carbonic anhydrase inhibitors.A failed tentative to design a super carbonic anhydrase having the biochemical properties of the most thermostable CA (SspCA) and the fastest (SazCA) enzymes.Protonography, a technique applicable for the analysis of η-carbonic anhydrase activity.Dithiocarbamates with potent inhibitory activity against the Saccharomyces cerevisiae β-carbonic anhydrase.Microbial Carbonic Anhydrases in Biomimetic Carbon Sequestration for Mitigating Global Warming: Prospects and Perspectives.Serendipitous fragment-based drug discovery: ketogenic diet metabolites and statins effectively inhibit several carbonic anhydrases.Polypharmacology of sulfonamides: pazopanib, a multitargeted receptor tyrosine kinase inhibitor in clinical use, potently inhibits several mammalian carbonic anhydrases.More effective dithiocarbamate derivatives inhibiting carbonic anhydrases, generated by QSAR and computational design.Molecular Docking and Anticonvulsant Activity of Newly Synthesized Quinazoline Derivatives.Discovery of curcumin inspired sulfonamide derivatives as a new class of carbonic anhydrase isoforms I, II, IX, and XII inhibitors.Sulfocoumarin-, Coumarin-, 4-Sulfamoylphenyl-Bearing Indazole-3-carboxamide Hybrids: Synthesis and Selective Inhibition of Tumor-Associated Carbonic Anhydrase Isozymes IX and XII.Anion inhibition studies of a beta carbonic anhydrase from the malaria mosquito Anopheles gambiae.Crystal structure of the human carbonic anhydrase II adduct with 1-(4-sulfamoylphenyl-ethyl)-2,4,6-triphenylpyridinium perchlorate, a membrane-impermeant, isoform selective inhibitor.Sulphonamide inhibition studies of the β-carbonic anhydrase from the bacterial pathogen Clostridium perfringens.A substituted sulfonamide and its Co (II), Cu (II), and Zn (II) complexes as potential antifungal agents.Synthesis and biological evaluation of dithiocarbamate esters of parthenolide as potential anti-acute myelogenous leukaemia agents
P2860
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P2860
Dithiocarbamates: a new class of carbonic anhydrase inhibitors. Crystallographic and kinetic investigations
description
2012 nî lūn-bûn
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2012 թուականի Փետրուարին հրատարակուած գիտական յօդուած
@hyw
2012 թվականի փետրվարին հրատարակված գիտական հոդված
@hy
2012年の論文
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2012年論文
@yue
2012年論文
@zh-hant
2012年論文
@zh-hk
2012年論文
@zh-mo
2012年論文
@zh-tw
2012年论文
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name
Dithiocarbamates: a new class ...... hic and kinetic investigations
@ast
Dithiocarbamates: a new class ...... hic and kinetic investigations
@en
Dithiocarbamates: a new class ...... hic and kinetic investigations
@nl
type
label
Dithiocarbamates: a new class ...... hic and kinetic investigations
@ast
Dithiocarbamates: a new class ...... hic and kinetic investigations
@en
Dithiocarbamates: a new class ...... hic and kinetic investigations
@nl
prefLabel
Dithiocarbamates: a new class ...... hic and kinetic investigations
@ast
Dithiocarbamates: a new class ...... hic and kinetic investigations
@en
Dithiocarbamates: a new class ...... hic and kinetic investigations
@nl
P2093
P2860
P50
P356
P1476
Dithiocarbamates: a new class ...... hic and kinetic investigations
@en
P2093
Alfonso Maresca
Fabrizio Carta
Mayank Aggarwal
P2860
P304
P356
10.1039/C2CC16395K
P407
P577
2012-02-11T00:00:00Z