Properly substituted analogues of BIX-01294 lose inhibition of G9a histone methyltransferase and gain selective anti-DNA methyltransferase 3A activity.
about
Polymyxins and quinazolines are LSD1/KDM1A inhibitors with unusual structural featuresEpigenetics in diagnosis, prognostic assessment and treatment of cancer: an update.DNA Methylation Targeting: The DNMT/HMT Crosstalk Challenge.Identification and optimization of hydrazone-gallate derivatives as specific inhibitors of DNA methyltransferase 3A.Identification of 2,4-diamino-6,7-dimethoxyquinoline derivatives as G9a inhibitors†Electronic supplementary information (ESI) available. See DOI: 10.1039/c4md00274a.Histone lysine methyltransferase structure activity relationships that allow for segregation of G9a inhibition and anti-Plasmodium activity† †The authors declare no competing interests. ‡ ‡Electronic supplementary information (ESI) available: SuppleHistone lysine methyltransferase structure activity relationships that allow for segregation of G9a inhibition and anti-Plasmodium activity.
P2860
Q28595992-10AA26F5-03E5-4F84-9B61-6B9BCE8D1AFAQ35726371-E0DB716E-0CA3-479A-8D57-FD7F34BAB3BCQ37729405-49B15F5A-9014-4C03-8659-12D07AE3EB88Q38786386-125E3CF0-0C58-4118-AADA-B841389974E6Q41269425-83734DB2-5715-4721-835F-A78B41665126Q47158353-24164465-DE70-426E-8B98-5BE5844393BFQ47200073-B8EC1EE1-9DAB-4269-869D-1E1E80FC91A7
P2860
Properly substituted analogues of BIX-01294 lose inhibition of G9a histone methyltransferase and gain selective anti-DNA methyltransferase 3A activity.
description
2014 nî lūn-bûn
@nan
2014 թուականի Մայիսին հրատարակուած գիտական յօդուած
@hyw
2014 թվականի մայիսին հրատարակված գիտական հոդված
@hy
2014年の論文
@ja
2014年論文
@yue
2014年論文
@zh-hant
2014年論文
@zh-hk
2014年論文
@zh-mo
2014年論文
@zh-tw
2014年论文
@wuu
name
Properly substituted analogues ...... methyltransferase 3A activity
@nl
Properly substituted analogues ...... methyltransferase 3A activity.
@ast
Properly substituted analogues ...... methyltransferase 3A activity.
@en
type
label
Properly substituted analogues ...... methyltransferase 3A activity
@nl
Properly substituted analogues ...... methyltransferase 3A activity.
@ast
Properly substituted analogues ...... methyltransferase 3A activity.
@en
prefLabel
Properly substituted analogues ...... methyltransferase 3A activity
@nl
Properly substituted analogues ...... methyltransferase 3A activity.
@ast
Properly substituted analogues ...... methyltransferase 3A activity.
@en
P2093
P2860
P50
P3181
P1433
P1476
Properly substituted analogues ...... methyltransferase 3A activity.
@en
P2093
Biagina Marrocco
Celine Bouvy
Christina Gros
Cindy Grandjenette
Domenico Tarantino
Donatella Labella
Fréderic Ausseil
Paola B Arimondo
Salvatore Di Maro
Valérie Poughon
P2860
P304
P3181
P356
10.1371/JOURNAL.PONE.0096941
P407
P577
2014-05-08T00:00:00Z