Promiscuous targeting of bromodomains by bromosporine identifies BET proteins as master regulators of primary transcription response in leukemia.
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Predictions of Ligand Selectivity from Absolute Binding Free Energy CalculationsDiscovery of a PCAF Bromodomain Chemical Probe.Identification of a Novel Class of BRD4 Inhibitors by Computational Screening and Binding Simulations.The bromodomain and extraterminal domain inhibitor bromosporine synergistically reactivates latent HIV-1 in latently infected cells.A theoretical insight into selectivity of inhibitors toward two domains of bromodomain-containing protein 4 using molecular dynamics simulations.Quantitative Characterization of Bivalent Probes for a Dual Bromodomain Protein, Transcription Initiation Factor TFIID Subunit 1.Activity of bromodomain protein inhibitors/binders against asexual-stage Plasmodium falciparum parasites.Large-scale analysis of water stability in bromodomain binding pockets with grand canonical Monte CarloDiscovery of a PCAF Bromodomain Chemical Probe
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Promiscuous targeting of bromodomains by bromosporine identifies BET proteins as master regulators of primary transcription response in leukemia.
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article científic
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article scientifique
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articolo scientifico
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artigo científico
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bilimsel makale
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scientific article published on 12 October 2016
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vedecký článok
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vetenskaplig artikel
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videnskabelig artikel
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vědecký článek
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name
Promiscuous targeting of bromo ...... cription response in leukemia.
@en
Promiscuous targeting of bromo ...... cription response in leukemia.
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type
label
Promiscuous targeting of bromo ...... cription response in leukemia.
@en
Promiscuous targeting of bromo ...... cription response in leukemia.
@nl
prefLabel
Promiscuous targeting of bromo ...... cription response in leukemia.
@en
Promiscuous targeting of bromo ...... cription response in leukemia.
@nl
P2093
P2860
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P356
P1433
P1476
Promiscuous targeting of bromo ...... scription response in leukemia
@en
P2093
Chen-Yi Wang
Cynthia Tallant
Hannah Lingard
Jean-Philippe Lambert
Juerg Schwaller
Katharina Leonards
Lucie Guetzoyan
Octovia Monteiro
Oliver Dovey
Sarah Picaud
P2860
P304
P356
10.1126/SCIADV.1600760
P50
P577
2016-10-12T00:00:00Z