Unprecedently Large-Scale Kinase Inhibitor Set Enabling the Accurate Prediction of Compound-Kinase Activities: A Way toward Selective Promiscuity by Design?
about
Computational-experimental approach to drug-target interaction mapping: A case study on kinase inhibitors.Progress towards a public chemogenomic set for protein kinases and a call for contributions.Kinome-Wide Profiling Prediction of Small Molecules.Beyond the hype: deep neural networks outperform established methods using a ChEMBL bioactivity benchmark set.Mapping of inhibitors and activity data to the human kinome and exploring promiscuity from a ligand and target perspective.Protocols for the Design of Kinase-Focused Compound Libraries.How to Achieve Better Results Using PASS-Based Virtual Screening: Case Study for Kinase Inhibitors.Clinical pharmacodynamic/exposure characterisation of the multikinase inhibitor ilorasertib (ABT-348) in a phase 1 dose-escalation trial.
P2860
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P2860
Unprecedently Large-Scale Kinase Inhibitor Set Enabling the Accurate Prediction of Compound-Kinase Activities: A Way toward Selective Promiscuity by Design?
description
2016 nî lūn-bûn
@nan
2016年の論文
@ja
2016年論文
@yue
2016年論文
@zh-hant
2016年論文
@zh-hk
2016年論文
@zh-mo
2016年論文
@zh-tw
2016年论文
@wuu
2016年论文
@zh
2016年论文
@zh-cn
name
Unprecedently Large-Scale Kina ...... lective Promiscuity by Design?
@en
Unprecedently Large-Scale Kina ...... lective Promiscuity by Design?
@nl
type
label
Unprecedently Large-Scale Kina ...... lective Promiscuity by Design?
@en
Unprecedently Large-Scale Kina ...... lective Promiscuity by Design?
@nl
prefLabel
Unprecedently Large-Scale Kina ...... lective Promiscuity by Design?
@en
Unprecedently Large-Scale Kina ...... lective Promiscuity by Design?
@nl
P2093
P2860
P50
P356
P1476
Unprecedently Large-Scale Kina ...... lective Promiscuity by Design?
@en
P2093
Alexander Roberts
Daniel Domine
Fanny Beltran Escudie
Serge Christmann-Franck
P2860
P304
P356
10.1021/ACS.JCIM.6B00122
P577
2016-08-02T00:00:00Z