Synthesis of peptide fluoromethyl ketones and the inhibition of human cathepsin B.
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Cysteine proteases as therapeutic targets: does selectivity matter? A systematic review of calpain and cathepsin inhibitorsDevelopment of Broad-Spectrum Halomethyl Ketone Inhibitors Against Coronavirus Main Protease 3CLproThe synthesis of lysylfluoromethanes and their properties as inhibitors of trypsin, plasmin and cathepsin BSynthesis and properties of peptidyl derivatives of arginylfluoromethanesThe synthesis of peptidylfluoromethanes and their properties as inhibitors of serine proteinases and cysteine proteinasesRetinoid-induced apoptosis and Sp1 cleavage occur independently of transcription and require caspase activationRecent developments in inhibiting cysteine and serine proteases.The specificity of bovine spleen cathepsin S. A comparison with rat liver cathepsins L and B.Antimalarial effects of peptide inhibitors of a Plasmodium falciparum cysteine proteinase.Suppression of Human T Cell Proliferation Mediated by the Cathepsin B Inhibitor, z-FA-FMK Is Due to Oxidative Stress.Role of Ced-3/ICE-family proteases in staurosporine-induced programmed cell death.Surface cathepsin B protects cytotoxic lymphocytes from self-destruction after degranulationCathepsin-B and cathepsin-L expression levels do not correlate with sensitivity of tumour cells to TNF-alpha-mediated apoptosis.Phorbol ester activation of a proteolytic cascade capable of activating latent transforming growth factor-betaL a process initiated by the exocytosis of cathepsin B.The cathepsin B inhibitor z-FA.fmk inhibits cytokine production in macrophages stimulated by lipopolysaccharide.Conditioned medium from ras oncogene-transformed NIH 3T3 cells induces bone resorption in vitro.The synthesis of arginylfluoroalkanes, their inhibition of trypsin and blood-coagulation serine proteinases and their anticoagulant activity.Design, synthesis and biological evaluation of a library of thiocarbazates and their activity as cysteine protease inhibitors.Release of cytochrome c and activation of pro-caspase-9 following lysosomal photodamage involves Bid cleavage.Cathepsin B regulates the intrinsic angiogenic threshold of endothelial cellsThe inactivation of the cysteinyl exopeptidases cathepsin H and C by affinity-labelling reagents.Comparative behaviour of calpain and cathepsin B toward peptidyl acyloxymethyl ketones, sulphonium methyl ketones and other potential inhibitors of cysteine proteinases.Pseudoarginine: synthesis and properties of derivatives of delta-(1-imidazolyl)norvaline.A role for caspases in lens fiber differentiationPeptidyl vinyl sulphones: a new class of potent and selective cysteine protease inhibitors: S2P2 specificity of human cathepsin O2 in comparison with cathepsins S and L.The cathepsin B inhibitor z-FA-CMK induces cell death in leukemic T cells via oxidative stress.Cloning of a cysteine protease required for the molting of Onchocerca volvulus third stage larvae.Exploring the interaction of some N-benzyloxycarbonyl-L-phenyl alanyl-L-alanine ketones and bovine spleen cathepsin B by molecular modeling and binding free energy calculation.
P2860
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P2860
Synthesis of peptide fluoromethyl ketones and the inhibition of human cathepsin B.
description
1985 nî lūn-bûn
@nan
1985年の論文
@ja
1985年論文
@yue
1985年論文
@zh-hant
1985年論文
@zh-hk
1985年論文
@zh-mo
1985年論文
@zh-tw
1985年论文
@wuu
1985年论文
@zh
1985年论文
@zh-cn
name
Synthesis of peptide fluoromethyl ketones and the inhibition of human cathepsin B.
@en
Synthesis of peptide fluoromethyl ketones and the inhibition of human cathepsin B.
@nl
type
label
Synthesis of peptide fluoromethyl ketones and the inhibition of human cathepsin B.
@en
Synthesis of peptide fluoromethyl ketones and the inhibition of human cathepsin B.
@nl
prefLabel
Synthesis of peptide fluoromethyl ketones and the inhibition of human cathepsin B.
@en
Synthesis of peptide fluoromethyl ketones and the inhibition of human cathepsin B.
@nl
P1476
Synthesis of peptide fluoromethyl ketones and the inhibition of human cathepsin B.
@en
P2093
P304
P356
10.1016/0003-2697(85)90598-6
P407
P577
1985-09-01T00:00:00Z