10-iodo-11H-indolo[3,2-c]quinoline-6-carboxylic acids are selective inhibitors of DYRK1A.
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Selectivity Profiling and Biological Activity of Novel β-Carbolines as Potent and Selective DYRK1 Kinase InhibitorsStructural analysis of pathogenic mutations in the DYRK1A gene in patients with developmental disorders.Pharmacology of Modulators of Alternative Splicing.DYRK1A inhibition as potential treatment for Alzheimer's disease.Synthesis of quinolines via copper-catalyzed domino reactions of enaminones.Molecular structures of cdc2-like kinases in complex with a new inhibitor chemotype.
P2860
10-iodo-11H-indolo[3,2-c]quinoline-6-carboxylic acids are selective inhibitors of DYRK1A.
description
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name
10-iodo-11H-indolo[3,2-c]quinoline-6-carboxylic acids are selective inhibitors of DYRK1A.
@en
10-iodo-11H-indolo[3,2-c]quinoline-6-carboxylic acids are selective inhibitors of DYRK1A.
@nl
type
label
10-iodo-11H-indolo[3,2-c]quinoline-6-carboxylic acids are selective inhibitors of DYRK1A.
@en
10-iodo-11H-indolo[3,2-c]quinoline-6-carboxylic acids are selective inhibitors of DYRK1A.
@nl
prefLabel
10-iodo-11H-indolo[3,2-c]quinoline-6-carboxylic acids are selective inhibitors of DYRK1A.
@en
10-iodo-11H-indolo[3,2-c]quinoline-6-carboxylic acids are selective inhibitors of DYRK1A.
@nl
P2093
P2860
P50
P356
P1476
10-iodo-11H-indolo[3,2-c]quinoline-6-carboxylic acids are selective inhibitors of DYRK1A.
@en
P2093
Anja Becker
Apirat Chaikuad
Conrad Kunick
Hannes Falke
Laurent Meijer
Nadège Loaëc
Olivier Lozach
Peter G Jones
Samira Abu Jhaisha
P2860
P304
P356
10.1021/JM501994D
P407
P577
2015-03-23T00:00:00Z