An Analog of BIX-01294 Selectively Inhibits a Family of Histone H3 Lysine 9 Jumonji Demethylases
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The role of histone demethylases in cancer therapyProperly substituted analogues of BIX-01294 lose inhibition of G9a histone methyltransferase and gain selective anti-DNA methyltransferase 3A activity.Modulation of epigenetic targets for anticancer therapy: clinicopathological relevance, structural data and drug discovery perspectivesTargeting histone lysine demethylases - progress, challenges, and the futureMiR137 is an androgen regulated repressor of an extended network of transcriptional coregulators.Identification of small molecule modulators of gene transcription with anticancer activity.Small-molecular modulators of cancer-associated epigenetic mechanisms.A small molecule modulates Jumonji histone demethylase activity and selectively inhibits cancer growth.Protein similarity networks reveal relationships among sequence, structure, and function within the Cupin superfamily.Pure Diastereomers of a Tranylcypromine-Based LSD1 Inhibitor: Enzyme Selectivity and In-Cell Studies.Inhibition of Nuclear Receptor Binding SET Domain 2/Multiple Myeloma SET Domain by LEM-06 Implication for Epigenetic Cancer Therapies.Successful strategies in the discovery of small-molecule epigenetic modulators with anticancer potential.Characterization of a Linked Jumonji Domain of the KDM5/JARID1 Family of Histone H3 Lysine 4 Demethylases.Quantitative analysis of histone demethylase probes using fluorescence polarizationStructural investigations of the nickel-induced inhibition of truncated constructs of the JMJD2 family of histone demethylases using X-ray absorption spectroscopy.Structural Basis for KDM5A Histone Lysine Demethylase Inhibition by Diverse CompoundsCurrent trends in epigenetic drug discovery.Lost in translation. New unexplored avenues for neuropsychopharmacology: epigenetics and microRNAs.JARID2 is a direct target of the PAX3-FOXO1 fusion protein and inhibits myogenic differentiation of rhabdomyosarcoma cells.Identification of 2,4-diamino-6,7-dimethoxyquinoline derivatives as G9a inhibitors†Electronic supplementary information (ESI) available. See DOI: 10.1039/c4md00274a.Epigenetic control and cancer: the potential of histone demethylases as therapeutic targets.Discovery of a Highly Selective Cell-Active Inhibitor of the Histone Lysine Demethylases KDM2/7.Pyrrole- and indole-containing tranylcypromine derivatives as novel lysine-specific demethylase 1 inhibitors active on cancer cellsDiscovery of a Highly Selective Cell-Active Inhibitor of the Histone Lysine Demethylases KDM2/7
P2860
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P2860
An Analog of BIX-01294 Selectively Inhibits a Family of Histone H3 Lysine 9 Jumonji Demethylases
description
2012 nî lūn-bûn
@nan
2012 թուականի Փետրուարին հրատարակուած գիտական յօդուած
@hyw
2012 թվականի փետրվարին հրատարակված գիտական հոդված
@hy
2012年の論文
@ja
2012年論文
@yue
2012年論文
@zh-hant
2012年論文
@zh-hk
2012年論文
@zh-mo
2012年論文
@zh-tw
2012年论文
@wuu
name
An Analog of BIX-01294 Selecti ...... Lysine 9 Jumonji Demethylases
@ast
An Analog of BIX-01294 Selecti ...... Lysine 9 Jumonji Demethylases
@en
An Analog of BIX-01294 Selecti ...... Lysine 9 Jumonji Demethylases
@nl
type
label
An Analog of BIX-01294 Selecti ...... Lysine 9 Jumonji Demethylases
@ast
An Analog of BIX-01294 Selecti ...... Lysine 9 Jumonji Demethylases
@en
An Analog of BIX-01294 Selecti ...... Lysine 9 Jumonji Demethylases
@nl
prefLabel
An Analog of BIX-01294 Selecti ...... Lysine 9 Jumonji Demethylases
@ast
An Analog of BIX-01294 Selecti ...... Lysine 9 Jumonji Demethylases
@en
An Analog of BIX-01294 Selecti ...... Lysine 9 Jumonji Demethylases
@nl
P2093
P2860
P50
P1476
An Analog of BIX-01294 Selecti ...... Lysine 9 Jumonji Demethylases
@en
P2093
Anup K Upadhyay
Donatella Labella
Ji Woong Han
Xiaodong Cheng
Xing Zhang
Young-Sup Yoon
P2860
P304
P356
10.1016/J.JMB.2011.12.036
P407
P577
2012-02-24T00:00:00Z