Irving Page Lecture: 5-HT(2A) serotonin receptor biology: interacting proteins, kinases and paradoxical regulation.
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Head-twitch response in rodents induced by the hallucinogen 2,5-dimethoxy-4-iodoamphetamine: a comprehensive history, a re-evaluation of mechanisms, and its utility as a model.DREADDs: novel tools for drug discovery and developmentA functional selectivity mechanism at the serotonin-2A GPCR involves ligand-dependent conformations of intracellular loop 2Fluorine in psychedelic phenethylaminesStructure-activity relationships of constrained phenylethylamine ligands for the serotonin 5-HT2 receptorsCannabinoid receptor agonists upregulate and enhance serotonin 2A (5-HT(2A)) receptor activity via ERK1/2 signaling.Sex hormones affect neurotransmitters and shape the adult female brain during hormonal transition periodsRole for serotonin2A (5-HT2A) and 2C (5-HT2C) receptors in experimental absence seizures.Cannabinoid 2 receptor- and beta Arrestin 2-dependent upregulation of serotonin 2A receptors.G-protein receptor kinase 5 regulates the cannabinoid receptor 2-induced up-regulation of serotonin 2A receptors.Cannabinoid-induced upregulation of serotonin 2A receptors in the hypothalamic paraventricular nucleus and anxiety-like behaviors in rats.Heterodimers of serotonin receptor subtypes 2 are driven by 5-HT2C protomers.Caveolin-1: Functional Insights into Its Role in Muscarine- and Serotonin-Induced Smooth Muscle Constriction in Murine Airways.Biochemistry. As good as chocolate.Metabotropic glutamate receptor 2 and corticotrophin-releasing factor receptor-1 gene expression is differently regulated by BDNF in rat primary cortical neurons.ERK is a Critical Regulator of JC Polyomavirus Infection.Synthesis, radiofluorination, and preliminary evaluation of the potential 5-HT2A receptor agonists [18 F]Cimbi-92 and [18 F]Cimbi-150.Serotonin receptors in hippocampusPathological Conditions Associated with the Disturbance of the 5-HT System
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Irving Page Lecture: 5-HT(2A) serotonin receptor biology: interacting proteins, kinases and paradoxical regulation.
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article científic
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article scientifique
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articolo scientifico
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artigo científico
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bilimsel makale
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scientific article published on February 2011
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vedecký článok
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vetenskaplig artikel
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videnskabelig artikel
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vědecký článek
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Irving Page Lecture: 5-HT(2A) ...... es and paradoxical regulation.
@en
Irving Page Lecture: 5-HT(2A) ...... es and paradoxical regulation.
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Irving Page Lecture: 5-HT(2A) ...... es and paradoxical regulation.
@en
Irving Page Lecture: 5-HT(2A) ...... es and paradoxical regulation.
@nl
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Irving Page Lecture: 5-HT(2A) ...... es and paradoxical regulation.
@en
Irving Page Lecture: 5-HT(2A) ...... es and paradoxical regulation.
@nl
P2860
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P1476
Irving Page Lecture: 5-HT(2A) ...... es and paradoxical regulation.
@en
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Bryan L Roth
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10.1016/J.NEUROPHARM.2011.01.012
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2011-02-01T00:00:00Z