In vitro and in vivo pharmacological characterization of the neuropeptide s receptor antagonist [D-Cys(tBu)5]neuropeptide S
about
Molecular evolution of the neuropeptide S receptorA novel brain penetrant NPS receptor antagonist, NCGC00185684, blocks alcohol-induced ERK-phosphorylation in the central amygdala and decreases operant alcohol self-administration in ratsIn vitro and in vivo pharmacological characterization of a neuropeptide S tetrabranched derivative.Abnormal response to stress and impaired NPS-induced hyperlocomotion, anxiolytic effect and corticosterone increase in mice lacking NPSR1.Behavioral phenotyping of neuropeptide S receptor knockout mice.Molecular fingerprint of neuropeptide S-producing neurons in the mouse brain.Neuropeptide S facilitates cue-induced relapse to cocaine seeking through activation of the hypothalamic hypocretin systemSelective Modulation of Gq/Gs pathways by Naphtho Pyrano Pyrimidines as antagonists of the Neuropeptide S Receptor.Synthesis and separation of the enantiomers of the neuropeptide S receptor antagonist (9R/S)-3-oxo-1,1-diphenyl-tetrahydro-oxazolo[3,4-a]pyrazine-7-carboxylic acid 4-fluoro-benzylamide (SHA 68).A single-nucleotide polymorphism of human neuropeptide s gene originated from Europe shows decreased bioactivityIntranasally administered neuropeptide S (NPS) exerts anxiolytic effects following internalization into NPS receptor-expressing neurons.Neuropeptide S: a novel regulator of pain-related amygdala plasticity and behaviorsFurther studies at neuropeptide s position 5: discovery of novel neuropeptide S receptor antagonistsNeuropeptide S: a transmitter system in the brain regulating fear and anxiety.Neuropeptide S receptor: recent updates on nonpeptide antagonist discovery.Neuropeptide S Induces Acute Anxiolysis by Phospholipase C-Dependent Signaling within the Medial Amygdala.Hypothalamic neuropeptide S receptor blockade decreases discriminative cue-induced reinstatement of cocaine seeking in the rat.Anxiolytic- and panicolytic-like effects of Neuropeptide S in the mouse elevated T-maze.Characterization of NGFFYamide Signaling in Starfish Reveals Roles in Regulation of Feeding Behavior and Locomotory Systems[d-Pen(p- t BuBzl)5]NPS, a novel ligand for the neuropeptide S receptor: structure activity and pharmacological studies
P2860
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P2860
In vitro and in vivo pharmacological characterization of the neuropeptide s receptor antagonist [D-Cys(tBu)5]neuropeptide S
description
2009 nî lūn-bûn
@nan
2009 թուականի Փետրուարին հրատարակուած գիտական յօդուած
@hyw
2009 թվականի փետրվարին հրատարակված գիտական հոդված
@hy
2009年の論文
@ja
2009年論文
@yue
2009年論文
@zh-hant
2009年論文
@zh-hk
2009年論文
@zh-mo
2009年論文
@zh-tw
2009年论文
@wuu
name
In vitro and in vivo pharmacol ...... st [D-Cys(tBu)5]neuropeptide S
@ast
In vitro and in vivo pharmacol ...... st [D-Cys(tBu)5]neuropeptide S
@en
In vitro and in vivo pharmacol ...... st [D-Cys(tBu)5]neuropeptide S
@nl
type
label
In vitro and in vivo pharmacol ...... st [D-Cys(tBu)5]neuropeptide S
@ast
In vitro and in vivo pharmacol ...... st [D-Cys(tBu)5]neuropeptide S
@en
In vitro and in vivo pharmacol ...... st [D-Cys(tBu)5]neuropeptide S
@nl
prefLabel
In vitro and in vivo pharmacol ...... st [D-Cys(tBu)5]neuropeptide S
@ast
In vitro and in vivo pharmacol ...... st [D-Cys(tBu)5]neuropeptide S
@en
In vitro and in vivo pharmacol ...... st [D-Cys(tBu)5]neuropeptide S
@nl
P2093
P2860
P50
P356
P1476
In vitro and in vivo pharmacol ...... st [D-Cys(tBu)5]neuropeptide S
@en
P2093
Anna Rizzi
Domenico Regoli
Girolamo Calò
Giuliano Marzola
Rainer K Reinscheid
Silvia Zucchini
Valeria Camarda
P2860
P304
P356
10.1124/JPET.108.143867
P407
P577
2009-02-01T00:00:00Z