Design, Synthesis, and Evaluation of Dibenzo[c,h][1,6]naphthyridines as Topoisomerase I Inhibitors and Potential Anticancer Agents
about
Exploring DNA topoisomerase I ligand space in search of novel anticancer agentsDesign, synthesis, and biological evaluation of O-2-modified indenoisoquinolines as dual topoisomerase I-tyrosyl-DNA phosphodiesterase I inhibitors.Dibenzo[c,h][1,5]naphthyridinediones as topoisomerase I inhibitors: design, synthesis, and biological evaluation.Design, Synthesis, and Biological Evaluation of Potential Prodrugs Related to the Experimental Anticancer Agent Indotecan (LMP400).Topoisomerase inhibitors as anticancer agents: a patent update.Microscopic Modes and Free Energies for Topoisomerase I-DNA Covalent Complex Binding with Non-campothecin Inhibitors by Molecular Docking and Dynamics Simulations.Quantitative structure-activity relationship studies on indenoisoquinoline topoisomerase I inhibitors as anticancer agents in human renal cell carcinoma cell line SN12C.Synthesis of indolo[4,3-bc]phenanthridine-6,11(2H,12H)-diones using the Schiff base-homophthalic anhydride cyclization reaction.Palladium meets copper: one-pot tandem synthesis of pyrido fused heterocycles via Sonogashira conjoined electrophilic cyclization.Iodine-catalyzed synthesis of dibenzo[b,h][1,6]naphthyridine-11-carboxamides via a domino reaction involving double elimination of hydrogen bromide.
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P2860
Design, Synthesis, and Evaluation of Dibenzo[c,h][1,6]naphthyridines as Topoisomerase I Inhibitors and Potential Anticancer Agents
description
2010 nî lūn-bûn
@nan
2010 թուականի Դեկտեմբերին հրատարակուած գիտական յօդուած
@hyw
2010 թվականի դեկտեմբերին հրատարակված գիտական հոդված
@hy
2010年の論文
@ja
2010年論文
@yue
2010年論文
@zh-hant
2010年論文
@zh-hk
2010年論文
@zh-mo
2010年論文
@zh-tw
2010年论文
@wuu
name
Design, Synthesis, and Evaluat ...... nd Potential Anticancer Agents
@ast
Design, Synthesis, and Evaluat ...... nd Potential Anticancer Agents
@en
type
label
Design, Synthesis, and Evaluat ...... nd Potential Anticancer Agents
@ast
Design, Synthesis, and Evaluat ...... nd Potential Anticancer Agents
@en
prefLabel
Design, Synthesis, and Evaluat ...... nd Potential Anticancer Agents
@ast
Design, Synthesis, and Evaluat ...... nd Potential Anticancer Agents
@en
P2093
P2860
P356
P1476
Design, Synthesis, and Evaluat ...... nd Potential Anticancer Agents
@en
P2093
Evgeny Kiselev
Mark Cushman
Thomas S. Dexheimer
P2860
P304
P356
10.1021/JM101048K
P407
P50
P577
2010-12-23T00:00:00Z