about
Pharmacophore Models and Pharmacophore-Based Virtual Screening: Concepts and Applications Exemplified on Hydroxysteroid DehydrogenasesSpecies used for drug testing reveal different inhibition susceptibility for 17beta-hydroxysteroid dehydrogenase type 1Hydroxybenzothiazoles as new nonsteroidal inhibitors of 17β-hydroxysteroid dehydrogenase type 1 (17β-HSD1)Focused libraries of 16-substituted estrone derivatives and modified e-ring steroids: inhibitors of 17beta-hydroxysteroid dehydrogenase type 1.Synthesis of libraries of 16beta-aminopropyl estradiol derivatives for targeting two key steroidogenic enzymes.Aromatase, estrone sulfatase, and 17β-hydroxysteroid dehydrogenase: structure-function studies and inhibitor development.Inhibitors of type 5 17β-hydroxysteroid dehydrogenase (AKR1C3): overview and structural insights.Perspectives in understanding the role of human 17beta-hydroxysteroid dehydrogenases in health and disease.The intraovarian actions of estrogen receptor-alpha are necessary to repress the formation of morphological and functional Leydig-like cells in the female gonad.Covalent Immobilization of Human Placental 17β-Hydroxysteroid Dehydrogenase Type 1 onto Glutaraldehyde Activated Silica Coupled with LC-TOF/MS for Anti-Cancer Drug Screening Applications.17beta-hydroxysteroid dehydrogenases in human breast cancer.17beta-Hydroxysteroid dehydrogenase inhibitors: a patent review.Human microsomal carbonyl reducing enzymes in the metabolism of xenobiotics: well-known and promising members of the SDR superfamily.Crucial Role of 3-Bromoethyl in Removing the Estrogenic Activity of 17β-HSD1 Inhibitor 16β-(m-Carbamoylbenzyl)estradiol.Predicting Putative Inhibitors of 17β-HSD1.Improved synthesis of EM-1745, preparation of its C17-ketone analogue and comparison of their inhibitory potency on 17beta-hydroxysteroid dehydrogenase type 1.17beta-hydroxysteroid dehydrogenase Type 1, and not Type 12, is a target for endocrine therapy of hormone-dependent breast cancer.Discovery of substituted 3-(phenylamino)benzoic acids as potent and selective inhibitors of type 5 17β-hydroxysteroid dehydrogenase (AKR1C3).Medical treatment improves social behavior in a primate endometriosis model (Callithrix jacchus).Identification of novel functional inhibitors of 17beta-hydroxysteroid dehydrogenase type III (17beta-HSD3).Inhibitors of type 1 17beta-hydroxysteroid dehydrogenase with reduced estrogenic activity: modifications of the positions 3 and 6 of estradiol.A 3D QSAR model of 17beta-HSD1 inhibitors based on a thieno[2,3-d]pyrimidin-4(3H)-one core applying molecular dynamics simulations and ligand-protein docking.Comparative investigation of the in vitro inhibitory potencies of 13-epimeric estrones and D-secoestrones towards 17β-hydroxysteroid dehydrogenase type 1.New inhibitors of fungal 17β-hydroxysteroid dehydrogenase based on the [1,5]-benzodiazepine scaffold
P2860
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P2860
description
2003 nî lūn-bûn
@nan
2003 թուականի Մարտին հրատարակուած գիտական յօդուած
@hyw
2003 թվականի մարտին հրատարակված գիտական հոդված
@hy
2003年の論文
@ja
2003年論文
@yue
2003年論文
@zh-hant
2003年論文
@zh-hk
2003年論文
@zh-mo
2003年論文
@zh-tw
2003年论文
@wuu
name
Inhibitors of 17 beta-hydroxysteroid dehydrogenases.
@ast
Inhibitors of 17 beta-hydroxysteroid dehydrogenases.
@en
Inhibitors of 17 beta-hydroxysteroid dehydrogenases.
@nl
type
label
Inhibitors of 17 beta-hydroxysteroid dehydrogenases.
@ast
Inhibitors of 17 beta-hydroxysteroid dehydrogenases.
@en
Inhibitors of 17 beta-hydroxysteroid dehydrogenases.
@nl
prefLabel
Inhibitors of 17 beta-hydroxysteroid dehydrogenases.
@ast
Inhibitors of 17 beta-hydroxysteroid dehydrogenases.
@en
Inhibitors of 17 beta-hydroxysteroid dehydrogenases.
@nl
P356
P1476
Inhibitors of 17 beta-hydroxysteroid dehydrogenases.
@en
P2093
Donald Poirier
P304
P356
10.2174/0929867033368222
P577
2003-03-01T00:00:00Z