Allosteric enhancers, allosteric agonists and ago-allosteric modulators: where do they bind and how do they act?
about
Flexible modulation of agonist efficacy at the human A3 adenosine receptor by the imidazoquinoline allosteric enhancer LUF6000Studies of the biogenic amine transporters. 13. Identification of "agonist" and "antagonist" allosteric modulators of amphetamine-induced dopamine releaseDrugs for allosteric sites on receptorsAllosteric Modulation of Sigma-1 Receptors Elicits Rapid Antidepressant ActivityText mining improves prediction of protein functional sites.Allosteric modulation of metabotropic glutamate receptors.Endogenous positive allosteric modulation of GABA(A) receptors by diazepam binding inhibitorSniffer patch laser uncaging response (SPLURgE): an assay of regional differences in allosteric receptor modulation and neurotransmitter clearanceInteractions of Cannabinoids With Biochemical SubstratesSeven transmembrane receptors as shapeshifting proteins: the impact of allosteric modulation and functional selectivity on new drug discovery.Teaching old receptors new tricks: biasing seven-transmembrane receptors.Mapping the druggable allosteric space of G-protein coupled receptors: a fragment-based molecular dynamics approach.Allosteric Modulation: An Alternate Approach Targeting the Cannabinoid CB1 Receptor.Agonist activation of alpha7 nicotinic acetylcholine receptors via an allosteric transmembrane siteGPR40 (FFAR1) - Combined Gs and Gq signaling in vitro is associated with robust incretin secretagogue action ex vivo and in vivoNovobiocin and peptide analogs of α-factor are positive allosteric modulators of the yeast G protein-coupled receptor Ste2p.Small molecules, peptides and natural products: getting a grip on 14-3-3 protein-protein modulation.L-Amino Acids Elicit Diverse Response Patterns in Taste Sensory Cells: A Role for Multiple Receptors.Structural dynamics and energetics underlying allosteric inactivation of the cannabinoid receptor CB1.Hunting for the function of orphan GPCRs - beyond the search for the endogenous ligand.Bioinformatics and variability in drug response: a protein structural perspective.Synaptic physiology of central CRH system.Studies of the biogenic amine transporters. 12. Identification of novel partial inhibitors of amphetamine-induced dopamine release.Growth hormone-releasing hormone as an agonist of the ghrelin receptor GHS-R1aML314: A Biased Neurotensin Receptor Ligand for Methamphetamine AbuseAllosteric modulators for the treatment of schizophrenia: targeting glutamatergic networksNovel 2- and 4-substituted 1H-imidazo[4,5-c]quinolin-4-amine derivatives as allosteric modulators of the A3 adenosine receptorQuinoline derivatives: candidate drugs for a class B G-protein coupled receptor, the calcitonin gene-related peptide receptor, a cause of migraines.Allosteric modulation of a cannabinoid G protein-coupled receptor: binding site elucidation and relationship to G protein signaling.Allosteric modulation of metabotropic glutamate receptors: structural insights and therapeutic potential.Novel GABA(B) receptor positive modulators: a patent survey.The changing world of G protein-coupled receptors: from monomers to dimers and receptor mosaics with allosteric receptor-receptor interactions.50th anniversary of the word "allosteric".Lifting the lid on GPCRs: the role of extracellular loops.Molecular alliance-from orthosteric and allosteric ligands to dualsteric/bitopic agonists at G protein coupled receptors.Quantitative analysis of receptor allosterism and its implication for drug discovery.Current status of A1 adenosine receptor allosteric enhancers.Preclinical Studies of Cannabinoid Reward, Treatments for Cannabis Use Disorder, and Addiction-Related Effects of Cannabinoid Exposure.Multivalent approaches and beyond: novel tools for the investigation of dopamine D2 receptor pharmacology.Biased agonism and allosteric modulation of G protein-coupled receptor 183 - a 7TM receptor also known as Epstein-Barr virus-induced gene 2.
P2860
Q21262008-FA7EA4B8-49B5-45DD-BD1F-73EBDA6CFB7CQ24655326-6D33C955-01D8-4DD5-BB9E-8D9F223FF8DEQ27006721-471EAE6D-942B-4381-9641-3B96A5B6DAD9Q28273055-3FDC09FE-7D0C-4340-B0DF-A7EB0D115795Q30413855-94B970B8-F819-419A-8498-4C2414759BDFQ30448534-D5F8AC67-23E7-4B45-A803-47F695175AC9Q30576168-27930BC6-D942-43DF-A8E5-7E47A51B1851Q33702403-673397A5-4C2C-4831-A9EE-9EB4F5678C4CQ33758351-36A85CB2-E248-4480-8937-B67F54475DECQ33890786-88124F4E-D7C3-4E00-8D92-271F23DD53CAQ33985759-27705917-C82F-49D4-8CDC-9312377A0A3FQ34054370-1BCB38C3-91BF-408D-87D0-3DB64CA1349BQ34545629-F157E7ED-62D7-4C05-8D16-945D527A5465Q34804573-2B5C76F0-216C-4BCD-9D41-3DAE6617D54DQ35040481-4EA983B1-30A4-4F6D-9305-B41D97C9C902Q35091488-EAD59635-6200-4023-94EE-730E984044CAQ35194362-FC2EFF8B-D158-4FA1-BE20-BEDEB9D9E22FQ35674119-7F77E676-9E79-4FC1-9E6D-61C288920D92Q35845768-12E51FE7-0F98-458A-B89E-424EE2A52B52Q35846184-3A952EC5-7ACE-40FD-8941-53953947D86FQ36009999-F87FEB24-2A22-473C-B891-0A58F81F724CQ36714050-2D381B07-2850-46B4-9594-D17DBB9B253FQ36926340-28513CFD-BFED-49EF-869D-D9723FDAB644Q37016373-803A4397-B490-4BD1-B256-49154E228EE3Q37099122-0EAB419E-4895-4CB3-AFF3-3CBD0AD53A46Q37220392-8FE3D29D-B172-4D32-A19D-2AA201F1D651Q37396368-EB73501E-DB38-4B4C-93BD-3E73B7DBDFB0Q37546168-CFA5C064-923C-418D-9FAC-EC8F8B232CE6Q37608491-EB90F6C3-2A25-424D-BDBF-9D6A9B4C6752Q37773480-838FED07-6830-4EAB-953E-B12532501CD9Q37774348-B17E075A-AFC1-4667-B1E6-BCCDE3C9D22BQ37777734-60F903E7-7653-4BEC-AA15-BEC2B7AD80A7Q37875827-14682866-98E9-414D-9E53-315B1C5C4010Q37921853-EB8AA43C-45DC-404F-8184-09FE39513901Q38066121-8BEDA5FF-D0A2-4ECF-BCC8-22CE842F3465Q38451155-F80CF0D5-51F5-4710-B2AD-F25B029AB633Q38542934-F8BB135D-9CAD-43E2-BC40-5556A24ED225Q38636791-08BA1D53-233D-4B48-A0DF-992D674A05C0Q38846984-D622E2E1-FC94-45D3-940A-4F862AE312E2Q38859909-97373C8B-551D-478B-9082-802B660AAC74
P2860
Allosteric enhancers, allosteric agonists and ago-allosteric modulators: where do they bind and how do they act?
description
2007 nî lūn-bûn
@nan
2007 թուականի Յուլիսին հրատարակուած գիտական յօդուած
@hyw
2007 թվականի հուլիսին հրատարակված գիտական հոդված
@hy
2007年の論文
@ja
2007年論文
@yue
2007年論文
@zh-hant
2007年論文
@zh-hk
2007年論文
@zh-mo
2007年論文
@zh-tw
2007年论文
@wuu
name
Allosteric enhancers, alloster ...... they bind and how do they act?
@ast
Allosteric enhancers, alloster ...... they bind and how do they act?
@en
Allosteric enhancers, alloster ...... they bind and how do they act?
@nl
type
label
Allosteric enhancers, alloster ...... they bind and how do they act?
@ast
Allosteric enhancers, alloster ...... they bind and how do they act?
@en
Allosteric enhancers, alloster ...... they bind and how do they act?
@nl
prefLabel
Allosteric enhancers, alloster ...... they bind and how do they act?
@ast
Allosteric enhancers, alloster ...... they bind and how do they act?
@en
Allosteric enhancers, alloster ...... they bind and how do they act?
@nl
P1476
Allosteric enhancers, alloster ...... they bind and how do they act?
@en
P304
P356
10.1016/J.TIPS.2007.06.008
P577
2007-07-13T00:00:00Z