In vivo regulation of monomer-tetramer conversion of pyruvate kinase subtype M2 by glucose is mediated via fructose 1,6-bisphosphate.
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Modulation of type M2 pyruvate kinase activity by the human papillomavirus type 16 E7 oncoproteinCancer Metabolism and Drug ResistanceThe Trypanocidal Drug Suramin and Other Trypan Blue Mimetics Are Inhibitors of Pyruvate Kinases and Bind to the Adenosine SitePyruvate kinase M2 activators promote tetramer formation and suppress tumorigenesisSmall Molecule Activation of PKM2 in Cancer Cells Induces Serine AuxotrophySerine is a natural ligand and allosteric activator of pyruvate kinase M2M2 pyruvate kinase provides a mechanism for nutrient sensing and regulation of cell proliferation.Metabolic reprogramming: a cancer hallmark even warburg did not anticipateDirect measurements of oscillatory glycolysis in pancreatic islet β-cells using novel fluorescence resonance energy transfer (FRET) biosensors for pyruvate kinase M2 activityPyruvate kinase type M2 promotes tumour cell exosome release via phosphorylating synaptosome-associated protein 23Three rounds (1R/2R/3R) of genome duplications and the evolution of the glycolytic pathway in vertebrates.Regulation of pyruvate metabolism and human diseasePyruvate kinase M2-specific siRNA induces apoptosis and tumor regressionQuinoline 3-sulfonamides inhibit lactate dehydrogenase A and reverse aerobic glycolysis in cancer cells.Pyruvate kinase M2 regulates gene transcription by acting as a protein kinase.Ca2+ Effects on ATP Production and Consumption Have Regulatory Roles on Oscillatory Islet Activity.Enhancing mitochondrial respiration suppresses tumor promoter TPA-induced PKM2 expression and cell transformation in skin epidermal JB6 cells.Reciprocal regulation of protein kinase and pyruvate kinase activities of pyruvate kinase M2 by growth signals.Regulation of thyroid hormone receptor-mediated transcription by a cytosol protein.Pyruvate kinase M2 regulates Hif-1α activity and IL-1β induction and is a critical determinant of the warburg effect in LPS-activated macrophages.Stress eating and tuning out: cancer cells re-wire metabolism to counter stress.Hallmarks of Pulmonary Hypertension: Mesenchymal and Inflammatory Cell Metabolic Reprogramming.Regulation of glycolysis in brown adipocytes by HIF-1αParkin Regulates the Activity of Pyruvate Kinase M2Human cytomegalovirus encoded chemokine receptor US28 activates the HIF-1α/PKM2 axis in glioblastoma cells.PKM2 inhibitor shikonin suppresses TPA-induced mitochondrial malfunction and proliferation of skin epidermal JB6 cells.PKM2, a Central Point of Regulation in Cancer Metabolism.A subunit interface mutant of yeast pyruvate kinase requires the allosteric activator fructose 1,6-bisphosphate for activityPyruvate Kinase Inhibits Proliferation during Postnatal Cerebellar Neurogenesis and Suppresses Medulloblastoma Formation.A Novel Role for Pyruvate Kinase M2 as a Corepressor for P53 during the DNA Damage Response in Human Tumor Cells.Glucose Catabolism in Liver Tumors Induced by c-MYC Can Be Sustained by Various PKM1/PKM2 Ratios and Pyruvate Kinase Activities.Pyruvate kinase M2 phosphorylates H2AX and promotes genomic instability in human tumor cells.Lapachol inhibits glycolysis in cancer cells by targeting pyruvate kinase M2.Oncogenic kinase-induced PKM2 tyrosine 105 phosphorylation converts non-oncogenic PKM2 to a tumor promoter and induces cancer stem-like cells.Posttranslational Modifications of Pyruvate Kinase M2: Tweaks that Benefit Cancer.Non-canonical functions of enzymes facilitate cross-talk between cell metabolic and regulatory pathways.An allostatic mechanism for M2 pyruvate kinase as an amino-acid sensor.
P2860
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P2860
In vivo regulation of monomer-tetramer conversion of pyruvate kinase subtype M2 by glucose is mediated via fructose 1,6-bisphosphate.
description
1991 nî lūn-bûn
@nan
1991 թուականի Սեպտեմբերին հրատարակուած գիտական յօդուած
@hyw
1991 թվականի սեպտեմբերին հրատարակված գիտական հոդված
@hy
1991年の論文
@ja
1991年論文
@yue
1991年論文
@zh-hant
1991年論文
@zh-hk
1991年論文
@zh-mo
1991年論文
@zh-tw
1991年论文
@wuu
name
In vivo regulation of monomer- ...... via fructose 1,6-bisphosphate.
@ast
In vivo regulation of monomer- ...... via fructose 1,6-bisphosphate.
@en
In vivo regulation of monomer- ...... via fructose 1,6-bisphosphate.
@nl
type
label
In vivo regulation of monomer- ...... via fructose 1,6-bisphosphate.
@ast
In vivo regulation of monomer- ...... via fructose 1,6-bisphosphate.
@en
In vivo regulation of monomer- ...... via fructose 1,6-bisphosphate.
@nl
prefLabel
In vivo regulation of monomer- ...... via fructose 1,6-bisphosphate.
@ast
In vivo regulation of monomer- ...... via fructose 1,6-bisphosphate.
@en
In vivo regulation of monomer- ...... via fructose 1,6-bisphosphate.
@nl
P2093
P1476
In vivo regulation of monomer- ...... via fructose 1,6-bisphosphate.
@en
P2093
Ashizawa K
Willingham MC
P304
16842-16846
P407
P577
1991-09-01T00:00:00Z