Structure-activity relationships of alpha-conotoxins targeting neuronal nicotinic acetylcholine receptors.
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Alpha7 nicotinic acetylcholine receptor is a target in pharmacology and toxicologyStructure of α-conotoxin BuIA: influences of disulfide connectivity on structural dynamicsRacemic and quasi-racemic X-ray structures of cyclic disulfide-rich peptide drug scaffoldsResidues Responsible for the Selectivity of α-Conotoxins for Ac-AChBP or nAChRsDietary breadth is positively correlated with venom complexity in cone snailsNMR and protein structure in drug design: application to cyclotides and conotoxins.Dockomatic - automated ligand creation and docking.Structure and activity of alpha-conotoxin PeIA at nicotinic acetylcholine receptor subtypes and GABA(B) receptor-coupled N-type calcium channelsAlanine scanning mutagenesis of the prototypic cyclotide reveals a cluster of residues essential for bioactivity.Alanine scan of α-conotoxin RegIIA reveals a selective α3β4 nicotinic acetylcholine receptor antagonist.Embryonic toxin expression in the cone snail Conus victoriae: primed to kill or divergent function?Molecular basis for the differential sensitivity of rat and human α9α10 nAChRs to α-conotoxin RgIA.Targeting the alpha9alpha10 nicotinic acetylcholine receptor to treat severe pain.Synthetic α-conotoxin mutants as probes for studying nicotinic acetylcholine receptors and in the development of novel drug leads.α-Conotoxins active at α3-containing nicotinic acetylcholine receptors and their molecular determinants for selective inhibition.Influence of disulfide connectivity on structure and bioactivity of α-conotoxin TxIA.DockoMatic: automated peptide analog creation for high throughput virtual screening.Inhibition of neuronal nicotinic acetylcholine receptor subtypes by alpha-Conotoxin GID and analogues.Alpha conotoxin-BuIA globular isomer is a competitive antagonist for oleoyl-L-alpha-lysophosphatidic acid binding to LPAR6; A molecular dynamics study.A novel α-conopeptide Eu1.6 inhibits N-type (CaV2.2) calcium channels and exhibits potent analgesic activity.Discovery of Peptide Drugs from Natural Sources
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P2860
Structure-activity relationships of alpha-conotoxins targeting neuronal nicotinic acetylcholine receptors.
description
2004 nî lūn-bûn
@nan
2004年の論文
@ja
2004年論文
@yue
2004年論文
@zh-hant
2004年論文
@zh-hk
2004年論文
@zh-mo
2004年論文
@zh-tw
2004年论文
@wuu
2004年论文
@zh
2004年论文
@zh-cn
name
Structure-activity relationshi ...... tinic acetylcholine receptors.
@ast
Structure-activity relationshi ...... tinic acetylcholine receptors.
@en
type
label
Structure-activity relationshi ...... tinic acetylcholine receptors.
@ast
Structure-activity relationshi ...... tinic acetylcholine receptors.
@en
prefLabel
Structure-activity relationshi ...... tinic acetylcholine receptors.
@ast
Structure-activity relationshi ...... tinic acetylcholine receptors.
@en
P2093
P2860
P1433
P1476
Structure-activity relationshi ...... tinic acetylcholine receptors.
@en
P2093
David J Craik
Emma L Millard
Norelle L Daly
P2860
P304
P356
10.1111/J.1432-1033.2004.04148.X
P407
P577
2004-06-01T00:00:00Z