Rigidified A3 Adenosine Receptor Agonists: 1-Deazaadenine Modification Maintains High in Vivo Efficacy
about
Metabolic mapping of A3 adenosine receptor agonist MRS5980Rigid Adenine Nucleoside Derivatives as Novel Modulators of the Human Sodium Symporters for Dopamine and Norepinephrine.A binding kinetics study of human adenosine A3 receptor agonists.Scaffold Repurposing of Nucleosides (Adenosine Receptor Agonists): Enhanced Activity at the Human Dopamine and Norepinephrine Sodium Symporters.Structure-Based Scaffold Repurposing for G Protein-Coupled Receptors: Transformation of Adenosine Derivatives into 5HT2B/5HT2C Serotonin Receptor Antagonists.Highly selective A3 adenosine receptor agonists relieve chronic neuropathic pain.Repurposing of a Nucleoside Scaffold from Adenosine Receptor Agonists to Opioid Receptor Antagonists
P2860
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P2860
Rigidified A3 Adenosine Receptor Agonists: 1-Deazaadenine Modification Maintains High in Vivo Efficacy
description
2015 nî lūn-bûn
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2015年の論文
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2015年論文
@yue
2015年論文
@zh-hant
2015年論文
@zh-hk
2015年論文
@zh-mo
2015年論文
@zh-tw
2015年论文
@wuu
2015年论文
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2015年论文
@zh-cn
name
Rigidified A3 Adenosine Recept ...... aintains High in Vivo Efficacy
@ast
Rigidified A3 Adenosine Recept ...... aintains High in Vivo Efficacy
@en
type
label
Rigidified A3 Adenosine Recept ...... aintains High in Vivo Efficacy
@ast
Rigidified A3 Adenosine Recept ...... aintains High in Vivo Efficacy
@en
prefLabel
Rigidified A3 Adenosine Recept ...... aintains High in Vivo Efficacy
@ast
Rigidified A3 Adenosine Recept ...... aintains High in Vivo Efficacy
@en
P2093
P2860
P50
P1476
Rigidified A3 Adenosine Recept ...... aintains High in Vivo Efficacy
@en
P2093
Daniela Salvemini
Elizabeth Gizewski
John A Auchampach
Steven Crane
Zhoumou Chen
P2860
P304
P356
10.1021/ACSMEDCHEMLETT.5B00150
P577
2015-05-20T00:00:00Z