Efficient, large-scale synthesis and preclinical studies of MRS5698, a highly selective A3 adenosine receptor agonist that protects against chronic neuropathic pain.
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Peripheral Adenosine A3 Receptor Activation Causes Regulated Hypothermia in Mice That Is Dependent on Central Histamine H1 Receptors.Purine (N)-Methanocarba Nucleoside Derivatives Lacking an Exocyclic Amine as Selective A3 Adenosine Receptor Agonists.Medicinal chemistry of adenosine, P2Y and P2X receptors.Cancer and orofacial pain.South (S)- and North (N)-Methanocarba-7-Deazaadenosine Analogues as Inhibitors of Human Adenosine Kinase.Scaffold Repurposing of Nucleosides (Adenosine Receptor Agonists): Enhanced Activity at the Human Dopamine and Norepinephrine Sodium Symporters.Structure-Based Scaffold Repurposing for G Protein-Coupled Receptors: Transformation of Adenosine Derivatives into 5HT2B/5HT2C Serotonin Receptor Antagonists.A Non-imaging High Throughput Approach to Chemical Library Screening at the Unmodified Adenosine-A3 Receptor in Living Cells.Pyrimidine Nucleotides Containing a (S)-Methanocarba Ring as P2Y6 Receptor Agonists.Chemotherapy-induced pain is promoted by enhanced spinal adenosine kinase levels via astrocyte-dependent mechanisms.Discovery of ERBB3 inhibitors for non-small cell lung cancer (NSCLC) via virtual screening.Repurposing of a Nucleoside Scaffold from Adenosine Receptor Agonists to Opioid Receptor Antagonists
P2860
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P2860
Efficient, large-scale synthesis and preclinical studies of MRS5698, a highly selective A3 adenosine receptor agonist that protects against chronic neuropathic pain.
description
2015 nî lūn-bûn
@nan
2015年の論文
@ja
2015年論文
@yue
2015年論文
@zh-hant
2015年論文
@zh-hk
2015年論文
@zh-mo
2015年論文
@zh-tw
2015年论文
@wuu
2015年论文
@zh
2015年论文
@zh-cn
name
Efficient, large-scale synthes ...... inst chronic neuropathic pain.
@ast
Efficient, large-scale synthes ...... inst chronic neuropathic pain.
@en
type
label
Efficient, large-scale synthes ...... inst chronic neuropathic pain.
@ast
Efficient, large-scale synthes ...... inst chronic neuropathic pain.
@en
prefLabel
Efficient, large-scale synthes ...... inst chronic neuropathic pain.
@ast
Efficient, large-scale synthes ...... inst chronic neuropathic pain.
@en
P2093
P2860
P1476
Efficient, large-scale synthes ...... inst chronic neuropathic pain.
@en
P2093
Daniela Salvemini
Janak Padia
Kenneth A Jacobson
P2860
P2888
P304
P356
10.1007/S11302-015-9459-2
P50
P577
2015-06-27T00:00:00Z