Characterizing the Covalent Targets of a Small Molecule Inhibitor of the Lysine Acetyltransferase P300.
about
The multifaceted role of lysine acetylation in cancer: prognostic biomarker and therapeutic targetEpigenetic Strategies to Boost Cancer Immunotherapies.Histone acetyltransferase inhibitors: where art thou?Inhibition of bromodomain and extra-terminal (BET) proteins increases NKG2D ligand MICA expression and sensitivity to NK cell-mediated cytotoxicity in multiple myeloma cells: role of cMYC-IRF4-miR-125b interplay.Assay interference and off-target liabilities of reported histone acetyltransferase inhibitors.CBP Regulates Recruitment and Release of Promoter-Proximal RNA Polymerase II.An AKAP-Lbc-RhoA interaction inhibitor promotes the translocation of aquaporin-2 to the plasma membrane of renal collecting duct principal cells.Discovery of Spiro Oxazolidinediones as Selective, Orally Bioavailable Inhibitors of p300/CBP Histone Acetyltransferases.Bioorthogonal pro-metabolites for profiling short chain fatty acylation.CREBBP/EP300 bromodomains are critical to sustain the GATA1/MYC regulatory axis in proliferation.Chemical Instability and Promiscuity of Arylmethylidenepyrazolinone-Based MDMX Inhibitors
P2860
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P2860
Characterizing the Covalent Targets of a Small Molecule Inhibitor of the Lysine Acetyltransferase P300.
description
2015 nî lūn-bûn
@nan
2015年の論文
@ja
2015年論文
@yue
2015年論文
@zh-hant
2015年論文
@zh-hk
2015年論文
@zh-mo
2015年論文
@zh-tw
2015年论文
@wuu
2015年论文
@zh
2015年论文
@zh-cn
name
Characterizing the Covalent Ta ...... Lysine Acetyltransferase P300.
@ast
Characterizing the Covalent Ta ...... Lysine Acetyltransferase P300.
@en
type
label
Characterizing the Covalent Ta ...... Lysine Acetyltransferase P300.
@ast
Characterizing the Covalent Ta ...... Lysine Acetyltransferase P300.
@en
prefLabel
Characterizing the Covalent Ta ...... Lysine Acetyltransferase P300.
@ast
Characterizing the Covalent Ta ...... Lysine Acetyltransferase P300.
@en
P2860
P50
P1476
Characterizing the Covalent Ta ...... Lysine Acetyltransferase P300.
@en
P2093
Julie M Garlick
Laura Guasch
P2860
P304
P356
10.1021/ACSMEDCHEMLETT.5B00385
P577
2015-10-31T00:00:00Z