Development of potent small-molecule inhibitors to drug the undruggable steroid receptor coactivator-3. - Wikidata - wikimedia - TriplyDB

Development of potent small-molecule inhibitors to drug the undruggable steroid receptor coactivator-3.

Development of potent small-molecule inhibitors to drug the undruggable steroid receptor coactivator-3.

http://www.wikidata.org/entity/Q37173140

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Targeting hepatic glucose metabolism in the treatment of type 2 diabetes.Estrogen receptor coregulator binding modulators (ERXs) effectively target estrogen receptor positive human breast cancers Molecular Pathways: Targeting Steroid Receptor Coactivators in Cancer.Dynamic contrast enhanced MRI detects changes in vascular transport rate constants following treatment with thermally-sensitive liposomal doxorubicin.Prognostic and predictive importance of the estrogen receptor coactivator AIB1 in a randomized trial comparing adjuvant letrozole and tamoxifen therapy in postmenopausal breast cancer: the Danish cohort of BIG 1-98.Coregulator profiling of the glucocorticoid receptor in lymphoid malignancies.Dynamic assembly and activation of estrogen receptor α enhancers through coregulator switching.Cancer Stem Cell Phenotypes in ER+ Breast Cancer Models are Promoted by PELP1/AIB1 Complexes.Targeting SRC Coactivators Blocks the Tumor-Initiating Capacity of Cancer Stem-like Cells.Chromatin reprogramming in breast cancer.Proteomic profiling identifies key coactivators utilized by mutant ERα proteins as potential new therapeutic targets.Steroid Receptor Coactivator-2 Controls the Pentose Phosphate Pathway through RPIA in Human Endometrial Cancer Cells

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Development of potent small-molecule inhibitors to drug the undruggable steroid receptor coactivator-3.

http://www.wikidata.org/entity/Q37173140

description

article científic

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article scientifique

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articolo scientifico

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artigo científico

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bilimsel makale

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scientific article published on 15 April 2016

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vedecký článok

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vetenskaplig artikel

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videnskabelig artikel

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vědecký článek

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name

Development of potent small-mo ...... teroid receptor coactivator-3.

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Development of potent small-mo ...... teroid receptor coactivator-3.

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type

label

Development of potent small-mo ...... teroid receptor coactivator-3.

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Development of potent small-mo ...... teroid receptor coactivator-3.

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prefLabel

Development of potent small-mo ...... teroid receptor coactivator-3.

@en

Development of potent small-mo ...... teroid receptor coactivator-3.

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PNAS.1604274113

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Proceedings of the National Academy of Sciences of the United States of America

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Development of potent small-mo ...... teroid receptor coactivator-3.

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Chengwei Zhang

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Dar-Chone Chow

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David M Lonard

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Jianming Xu

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Jianwei Chen

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Jin Wang

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Mingkun Zhao

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Timothy Palzkill

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Xianzhou Song

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Yang Yu

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P2860

Nuclear receptor coregulators: modulators of pathology and therapeutic targets

Crystal structure of the sodium-potassium pump (Na+,K+-ATPase) with bound potassium and ouabain

Sequence and characterization of a coactivator for the steroid hormone receptor superfamily

Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings

The atomic structure of protein-protein recognition sites

Identification of verrucarin a as a potent and selective steroid receptor coactivator-3 small molecule inhibitor

Fast Calculation of Molecular Polar Surface Area as a Sum of Fragment-Based Contributions and Its Application to the Prediction of Drug Transport Properties

Reaching for high-hanging fruit in drug discovery at protein-protein interfaces

Genes that mediate breast cancer metastasis to lung

A hot spot of binding energy in a hormone-receptor interface

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4970-4975

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scholarly article

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10.1073/PNAS.1604274113

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18

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113

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Bert W. O'Malley

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2016-04-15T00:00:00Z

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27084884

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4983835

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