The impact of assay technology as applied to safety assessment in reducing compound attrition in drug discovery.
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Biological detection by optical oxygen sensing.Stem cells and stem cell-derived tissues and their use in safety assessment.Toward predictive models for drug-induced liver injury in humans: are we there yet?Oncogenic protein interfaces: small molecules, big challenges.Mechanisms of amiodarone and valproic acid induced liver steatosis in mouse in vivo act as a template for other hepatotoxicity models.From Type I to Type II: Design, Synthesis, and Characterization of Potent Pyrazin-2-ones as DFG-Out Inhibitors of PDGFRβ.Phenotypic profiling of structural cardiotoxins in vitro reveals dependency on multiple mechanisms of toxicity.A testing strategy to predict risk for drug-induced liver injury in humans using high-content screen assays and the 'rule-of-two' model.How can we discover safer drugs?
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The impact of assay technology as applied to safety assessment in reducing compound attrition in drug discovery.
description
article científic
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article scientifique
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articol științific
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articolo scientifico
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artigo científico
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artigo científico
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artigo científico
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artikel ilmiah
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artikull shkencor
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artículo científico
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name
The impact of assay technology ...... d attrition in drug discovery.
@en
The impact of assay technology ...... d attrition in drug discovery.
@nl
type
label
The impact of assay technology ...... d attrition in drug discovery.
@en
The impact of assay technology ...... d attrition in drug discovery.
@nl
prefLabel
The impact of assay technology ...... d attrition in drug discovery.
@en
The impact of assay technology ...... d attrition in drug discovery.
@nl
P2860
P1476
The impact of assay technology ...... d attrition in drug discovery.
@en
P2093
Craig E Thomas
Yvonne Will
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P304
P356
10.1517/17460441.2012.651122
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P577
2012-01-09T00:00:00Z