Cathepsin B Inhibitors: Combining Dipeptide Nitriles with an Occluding Loop Recognition Element by Click Chemistry.

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Cathepsin B and L inhibitors: a patent review (2010 - present).Addition of 2-(ethylamino)acetonitrile group to nitroxoline results in significantly improved anti-tumor activity in vitro and in vivo

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Cathepsin B Inhibitors: Combining Dipeptide Nitriles with an Occluding Loop Recognition Element by Click Chemistry.

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Cathepsin B Inhibitors: Combin ...... on Element by Click Chemistry.

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Cathepsin B Inhibitors: Combin ...... on Element by Click Chemistry.

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Janina Schmitz

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Michael Gütschow

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Tianwei Li

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Ulrike Bartz

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P2860

L-trans-Epoxysuccinyl-leucylamido(4-guanidino)butane (E-64) and its analogues as inhibitors of cysteine proteinases including cathepsins B, H and L

Cysteine cathepsins: their role in tumor progression and recent trends in the development of imaging probes

Identification of dipeptidyl nitriles as potent and selective inhibitors of cathepsin B through structure-based drug design

The refined 2.15 A X-ray crystal structure of human liver cathepsin B: the structural basis for its specificity

Novel mechanism of cathepsin B inhibition by antibiotic nitroxoline and related compounds

Development of N-(Functionalized benzoyl)-homocycloleucyl-glycinonitriles as Potent Cathepsin K Inhibitors

Crystal structure of cathepsin B inhibited with CA030 at 2.0-A resolution: A basis for the design of specific epoxysuccinyl inhibitors

Redox-based inactivation of cysteine cathepsins by compounds containing the 4-aminophenol moiety

Azapeptides structurally based upon inhibitory sites of cystatins as potent and selective inhibitors of cysteine proteases.

A double-headed cathepsin B inhibitor devoid of warhead.

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scholarly article

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10.1021/ACSMEDCHEMLETT.5B00474

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Cathepsin B Inhibitors: Combining Dipeptide Nitriles with an Occluding Loop Recognition Element by Click Chemistry.

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P2860

Cathepsin B Inhibitors: Combining Dipeptide Nitriles with an Occluding Loop Recognition Element by Click Chemistry.

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