Dermorphin gene sequence peptide with high affinity and selectivity for delta-opioid receptors.
about
6-N,N-dimethylamino-2,3-naphthalimide: a new environment-sensitive fluorescent probe in delta- and mu-selective opioid peptides.Further studies on lead compounds containing the opioid pharmacophore Dmt-Tic.cDNAs encoding [D-Ala2]deltorphin precursors from skin of Phyllomedusa bicolor also contain genetic information for three dermorphin-related opioid peptides.Role of 2',6'-dimethyl-l-tyrosine (Dmt) in some opioid lead compoundsNew 2',6'-dimethyl-L-tyrosine (Dmt) opioid peptidomimetics based on the Aba-Gly scaffold. Development of unique mu-opioid receptor ligandsFrog skin opioid peptides: a case for environmental mimicry.Opioid activity of dermenkephalin analogues in the guinea-pig myenteric plexus and the hamster vas deferens.A new opioid designed multiple ligand derived from the micro opioid agonist endomorphin-2 and the delta opioid antagonist pharmacophore Dmt-TicDelta opioidmimetic antagonists: prototypes for designing a new generation of ultraselective opioid peptides.Design and synthesis of opioidmimetics containing 2',6'-dimethyl-L-tyrosine and a pyrazinone-ring platform.Further studies on the effect of lysine at the C-terminus of the Dmt-Tic opioid pharmacophore.Role of benzimidazole (Bid) in the delta-opioid agonist pseudopeptide H-Dmt-Tic-NH-CH(2)-Bid (UFP-502)Effect of lysine at C-terminus of the Dmt-Tic opioid pharmacophore.Synthesis of 3,6-bis[H-Tyr/H-Dmt-NH(CH2)m,n]-2(1H)pyrazinone derivatives: function of alkyl chain length on opioid activity.Synthesis of a potent and selective (18)F-labeled delta-opioid receptor antagonist derived from the Dmt-Tic pharmacophore for positron emission tomography imaging.
P2860
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P2860
Dermorphin gene sequence peptide with high affinity and selectivity for delta-opioid receptors.
description
1989 nî lūn-bûn
@nan
1989年の論文
@ja
1989年学术文章
@wuu
1989年学术文章
@zh-cn
1989年学术文章
@zh-hans
1989年学术文章
@zh-my
1989年学术文章
@zh-sg
1989年學術文章
@yue
1989年學術文章
@zh
1989年學術文章
@zh-hant
name
Dermorphin gene sequence pepti ...... ty for delta-opioid receptors.
@en
type
label
Dermorphin gene sequence pepti ...... ty for delta-opioid receptors.
@en
prefLabel
Dermorphin gene sequence pepti ...... ty for delta-opioid receptors.
@en
P2093
P1476
Dermorphin gene sequence pepti ...... ty for delta-opioid receptors.
@en
P2093
A Guglietta
L H Lazarus
R de Castiglione
W E Wilson
P304
P407
P577
1989-02-01T00:00:00Z