about
Cyclohexylcarbamic acid 3'- or 4'-substituted biphenyl-3-yl esters as fatty acid amide hydrolase inhibitors: synthesis, quantitative structure-activity relationships, and molecular modeling studiesNew family of polyamine macrocycles containing 2,5-diphenyl[1,3,4]oxadiazole as a signaling unit. Synthesis, acid-base and spectrophotometric properties.Design, synthesis, and structure-activity relationships of alkylcarbamic acid aryl esters, a new class of fatty acid amide hydrolase inhibitors.Divergent synthesis of novel 9-deazaxanthine derivatives via late-stage cross-coupling reactions.Synthesis and quantitative structure-activity relationship of fatty acid amide hydrolase inhibitors: modulation at the N-portion of biphenyl-3-yl alkylcarbamates.Enantioselective total synthesis of (-)-acylfulvene and (-)-irofulven.Observations in the Synthesis of the Core of the Antitumor Illudins via an Enyne Ring Closing Metathesis CascadeSynthesis of 2-substituted tryptophans via a C3- to C2-alkyl migration.A novel one-pot approach of hexahydropyrrolo[2,3-b]indole nucleus by a cascade addition/cyclization strategy: synthesis of (+/-)-esermethole.Direct B-alkyl Suzuki-Miyaura cross-coupling of 2-halopurines. Practical synthesis of ST1535, a potent adenosine A2A receptor antagonist.Diastereo- and enantioselective hydrogenation of a challenging enamide derived from 4-phenyl-2-tetralone: an appealing shortcut towards enantiopure cis-2-aminotetraline derivatives.Conformation by NMR of two tetralin-based receptor ligands.Synthesis and biological evaluation of metabolites of 2-n-butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine (ST1535), a potent antagonist of the A2A adenosine receptor for the treatment of Parkinson's disease.Tricyclic alkylamides as melatonin receptor ligands with antagonist or inverse agonist activity.Synthesis of (E)-8-(3-chlorostyryl)caffeine analogues leading to 9-deazaxanthine derivatives as dual A(2A) antagonists/MAO-B inhibitors.Synthesis of (-)-epi-indolactam V by an intramolecular Buchwald-Hartwig C-N coupling cyclization reaction.Switchable reactivity of acylated alpha, beta-dehydroamino ester in the Friedel-Crafts alkylation of indoles by changing the Lewis acid.An improved synthesis of cis-4-phenyl-2-propionamidotetralin (4-P-PDOT): a selective MT(2) melatonin receptor antagonist.Synthesis of benzo[1,2-d;3,4-d']diimidazole and 1H-pyrazolo[4,3-b]pyridine as putative A2A receptor antagonists.Iron-Catalyzed Direct C3-Benzylation of Indoles with Benzyl Alcohols through Borrowing Hydrogen.Iridium-catalyzed direct synthesis of tryptamine derivatives from indoles: exploiting n-protected β-amino alcohols as alkylating agents.Palladium(II)-Catalyzed Intramolecular Oxidative C-H/C-H Cross-Coupling Reaction of C3,N-Linked Biheterocycles: Rapid Access to Polycyclic Nitrogen Heterocycles.Palladium(II)-Catalyzed Cross-Dehydrogenative Coupling (CDC) of N-Phthaloyl Dehydroalanine Esters with Simple Arenes: Stereoselective Synthesis of Z-Dehydrophenylalanine Derivatives.Synthesis and configuration determination of all enantiopure stereoisomers of the melatonin receptor ligand 4-phenyl-2-propionamidotetralin using an expedient optical resolution of 4-phenyl-2-tetralone.Organocatalytic Aza-Friedel-Crafts/Lactonization Domino Reaction of Naphthols and Phenols with 2-Acetamidoacrylate to Naphtho- and Benzofuranones Bearing a Quaternary Center at the C3 PositionNew branched macrocyclic ligand and its side-arm, two urea-based receptors for anions: synthesis, binding studies and crystal structureSynthesis of Tryptamine Derivatives via a Direct, One-Pot Reductive Alkylation of IndolesDirect, One-Pot Reductive Alkylation of Anilines with Functionalized Acetals Mediated by Triethylsilane and TFA. Straightforward Route for Unsymmetrically Substituted EthylenediamineThe collisional behavior of ESI-generated protonated molecules of some carbamate FAAH inhibitors isosteres and its relationships with biological activityCorrelation between energetics of collisionally activated decompositions, interaction energy and biological potency of carbamate FAAH inhibitorsSynthesis and Structure-Activity Relationships of FAAH Inhibitors: Cyclohexylcarbamic Acid Biphenyl Esters with Chemical Modulation at the Proximal Phenyl RingEnantioselective total synthesis of (-)-acylfulvene and (-)-irofulvenFacile synthesis of @-tide beta-strand peptidomimetics: improved assembly in solution and on solid phaseDirect preparation of unsymmetrical difunctionalized cyclen derivatives by an Ugi multicomponent reactionDirect, regioselective, and chemoselective preparation of novel boronated tryptophans by Friedel-Crafts alkylationPotent, Metabolically Stable 2-Alkyl-8-(2H-1,2,3-triazol-2-yl)-9H-adenines as Adenosine A2A Receptor LigandsSynthesis of (±)-cis-clavicipitic acid by a Rh(I)-catalyzed intramolecular imine reactionA simple, modular synthesis of C4-substituted tryptophan derivativesTotal Synthesis of (-)-Clavicipitic Acid via γ,γ-Dimethylallyltryptophan (DMAT) and Chemoselective C-H HydroxylationConcise and Convergent Enantioselective Total Syntheses of (+)- and (-)-Fumimycin
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Q28285285-8D5D1A3F-9987-4F94-B529-7DA25F13C2A7Q33537196-84C50E61-4EC0-46C4-ADB3-E1DDC2F42165Q34200866-21415F80-100B-40E0-B19D-4B73269629B9Q34437316-082D7CEC-22F8-4743-A21D-7B05FC2F2349Q37098652-66A8D123-841A-4634-B63B-8F46A6ED742EQ41865123-63F31521-5114-4D52-90A3-297FA1756139Q42590408-E5E5E12E-1EE3-463C-8168-6E6EE61E3438Q42906265-7C444D91-B280-4767-AC31-44EF6A2D980DQ42925125-2693AC6F-523E-4958-A7CA-E94B97A9A7AEQ42992320-13FBC2E4-0FFF-4B23-AC4E-28B2B68A3E3AQ43182193-95B744D9-78B9-40CD-8AE0-58F4925B44E4Q44485803-4F1BF5D8-E459-4A7C-AE26-54888548DABCQ44587073-0A1EE83B-7CC6-4148-95F9-9C7458767507Q45007066-7FCBAA24-6065-4466-BD8A-4EEC237A0530Q46076494-7C0BADC2-DE48-4D7F-B677-0F9AD191C58EQ46475372-CFD2E1E8-79E1-4EEB-8FB5-A041A63A07F6Q46536268-A5E5D710-9E6F-494B-82E3-5865519510B9Q46853883-AAE16621-43E7-459A-870A-2C0F690EDBF3Q46895554-ADF71997-17B4-4E33-AE5A-721F6B8668F5Q48343285-336A0DA1-062D-4BB5-9A7F-11EB4FA6CBC2Q51006460-997DA846-C962-45DB-A40E-4E66868896F8Q52750915-13D53987-2E93-422B-9217-B469C8D9A0AAQ52868270-6F25E177-E277-498B-BB31-E8A192E08F27Q53204974-A99AB08A-44A5-4A2E-AE0F-DD8C4F5F10A9Q56983278-2AC263FA-C8EF-45BF-835C-DC9CA73081B9Q60257297-FB20ABF1-F96E-4D2B-BCBE-F7559AA5917EQ61781545-15206130-7078-4581-9FF0-F54E3ED62EB9Q61781548-36FFBE58-E672-4FD4-BC92-10AB66ADC9B9Q63423448-9F070342-7A1A-440A-A137-B1E9794A1195Q63423520-C68DF8F5-4191-4D4C-8165-5E0765104130Q63423653-81EAA5E8-F27F-46A2-8B88-6BE8A953F482Q80059589-AA818068-A9D0-4AAC-85DA-47005A10B69DQ81017392-713207C3-68EB-4863-BA81-0A5877B55A52Q83007726-AEB3AD77-9777-4B79-AD80-B0899AB87424Q83156893-BD91CEEA-9314-4085-B75C-C9EEAF8EAE54Q87262241-D0CAC1D6-6ECB-4CE5-AAA9-E7CFCA24163AQ87413382-A43BDB55-A4FC-42C1-B856-725318B14D59Q88521589-311F8209-3D95-4F2A-8A8D-D01513869940Q92236857-E3B30CFE-0D07-45F4-A607-6D958943DD7AQ93058828-82364AB1-7FA1-44AF-B01E-471536E21055
P50
description
hulumtues
@sq
researcher
@en
wetenschapper
@nl
հետազոտող
@hy
name
Giovanni Piersanti
@ast
Giovanni Piersanti
@en
Giovanni Piersanti
@es
Giovanni Piersanti
@nl
Giovanni Piersanti
@sl
type
label
Giovanni Piersanti
@ast
Giovanni Piersanti
@en
Giovanni Piersanti
@es
Giovanni Piersanti
@nl
Giovanni Piersanti
@sl
prefLabel
Giovanni Piersanti
@ast
Giovanni Piersanti
@en
Giovanni Piersanti
@es
Giovanni Piersanti
@nl
Giovanni Piersanti
@sl
P108
P1053
E-1656-2015
P106
P1153
6602863677
P21
P31
P3829
P496
0000-0003-0418-7143