Control of conformational equilibria in the human B2 bradykinin receptor. Modeling of nonpeptidic ligand action and comparison to the rhodopsin structure.

Control of conformational equilibria in the human B2 bradykinin receptor. Modeling of nonpeptidic ligand action and comparison to the rhodopsin structure.

Item
http://www.wikidata.org/entity/Q43701636
Identification by site-directed mutagenesis of residues involved in ligand recognition and activation of the human A3 adenosine receptor.The crystallographic model of rhodopsin and its use in studies of other G protein-coupled receptors.New insights into the stereochemical requirements of the bradykinin B2 receptor antagonists binding.Pharmacological characterization of ligand-receptor interactions at the zebrafish bradykinin receptor.Effect of a toggle switch mutation in TM6 of the human adenosine A₃ receptor on Gi protein-dependent signalling and Gi-independent receptor internalization.A conserved aromatic lock for the tryptophan rotameric switch in TM-VI of seven-transmembrane receptors.Conserved helix 7 tyrosine acts as a multistate conformational switch in the 5HT2C receptor. Identification of a novel "locked-on" phenotype and double revertant mutations.Comparison of the molecular interactions of two antagonists, MEN16132 or icatibant, at the human kinin B₂ receptor.A different molecular interaction of bradykinin and the synthetic agonist FR190997 with the human B2 receptor: evidence from mutational analysis.Preliminary mutational analysis of the human kinin B2 receptor for nonpeptide antagonist ligands recognition.Agonist-specific transactivation of phosphoinositide 3-kinase signaling pathway mediated by the dopamine D2 receptor.Comparative analysis of putative agonist-binding modes in the human A1 adenosine receptor.Optical biosensor provides insights for bradykinin B(2) receptor signaling in A431 cells.Dual antagonists of the bradykinin B1 and B2 receptors based on a postulated common pharmacophore from existing non-peptide antagonists.
P2860

Control of conformational equilibria in the human B2 bradykinin receptor. Modeling of nonpeptidic ligand action and comparison to the rhodopsin structure.

Item
http://www.wikidata.org/entity/Q43701636
description
2001 nî lūn-bûn
@nan
2001年の論文
@ja
2001年学术文章
@wuu
2001年学术文章
@zh
2001年学术文章
@zh-cn
2001年学术文章
@zh-hans
2001年学术文章
@zh-my
2001年学术文章
@zh-sg
2001年學術文章
@yue
2001年學術文章
@zh-hant
name
Control of conformational equi ...... on to the rhodopsin structure.
@en
Control of conformational equi ...... on to the rhodopsin structure.
@nl
type
label
Control of conformational equi ...... on to the rhodopsin structure.
@en
Control of conformational equi ...... on to the rhodopsin structure.
@nl
prefLabel
Control of conformational equi ...... on to the rhodopsin structure.
@en
Control of conformational equi ...... on to the rhodopsin structure.
@nl
P1433
P1476
P2093
P2860
P304
P31
P356
P407
P433
P478
P50
P577
P698
P356
P1433
P1476
Control of conformational equi ...... son to the rhodopsin structure
@en
P2093
P2860
P304
P31
P356
P407
P433
P478
P50
P577
P698