about
Suppression of the hypothalamic-pituitary-gonadal axis by TAK-385 (relugolix), a novel, investigational, orally active, small molecule gonadotropin-releasing hormone (GnRH) antagonist: studies in human GnRH receptor knock-in mice.The RNA helicase DDX39B and its paralog DDX39A regulate androgen receptor splice variant AR-V7 generation.Glycogen synthase kinase-3 inhibitors suppress the AR-V7-mediated transcription and selectively inhibit cell growth in AR-V7-positive prostate cancer cells.Retinal neuronal death induced by intraocular administration of a nitric oxide donor and its rescue by neurotrophic factors in rats.Neuronal nitric oxide synthase is crucial for ganglion cell death in rat retinal explant cultures.A novel androgen-dependent prostate cancer xenograft model derived from skin metastasis of a Japanese patient.Evaluation of pharmacokinetics/pharmacodynamics and efficacy of one-month depots of TAK-448 and TAK-683, investigational kisspeptin analogs, in male rats and an androgen-dependent prostate cancer model.Discovery of Novel 5-(Piperazine-1-carbonyl)pyridin-2(1H)-one Derivatives as Orally eIF4A3-Selective Inhibitors.Growth Inhibition by Testosterone in an Androgen Receptor Splice Variant-Driven Prostate Cancer Model.Pharmacologic profiles of investigational kisspeptin/metastin analogues, TAK-448 and TAK-683, in adult male rats in comparison to the GnRH analogue leuprolide.CDK8/19 inhibition induces premature G1/S transition and ATR-dependent cell death in prostate cancer cells.Anti-tumor efficacy of a novel CLK inhibitor via targeting RNA splicing and MYC-dependent vulnerability.
P50
Q34391535-7A9797EC-816A-45E4-80F2-659794FA9AF9Q36233615-BFE1D9ED-EC78-4C33-A8E7-8F2C1CE041CBQ38708121-98197C0A-7749-41D7-B350-866DCFEAF216Q44376479-16DA6D07-14EF-47BD-B371-E64F0DADCD4FQ44743525-19F41C35-1E9B-4105-ADDB-AFE668881FD4Q45915275-813A4A3B-8B9C-467A-AD43-155E0376B84FQ49885502-AD943A30-7447-4B08-A114-D475F6F81B53Q50066105-56F37A9D-F10B-4D82-A90A-4734FC2BC08CQ51606183-CB949BC1-E7D8-49E5-A624-A73553AC9912Q51749160-E3B1431A-2154-4998-A142-1896A597E751Q52345436-314EA841-D933-4EDA-8FAD-8851F6D5512AQ54978916-AECC0258-5309-4DA6-BEA1-58488511556A
P50
description
hulumtues
@sq
researcher
@en
wetenschapper
@nl
հետազոտող
@hy
name
Daisuke Nakata
@ast
Daisuke Nakata
@en
Daisuke Nakata
@es
Daisuke Nakata
@nl
Daisuke Nakata
@sl
type
label
Daisuke Nakata
@ast
Daisuke Nakata
@en
Daisuke Nakata
@es
Daisuke Nakata
@nl
Daisuke Nakata
@sl
prefLabel
Daisuke Nakata
@ast
Daisuke Nakata
@en
Daisuke Nakata
@es
Daisuke Nakata
@nl
Daisuke Nakata
@sl
P106
P21
P31
P496
0000-0002-7891-2275