Miniaturized receptor binding assays: complications arising from ligand depletion.
about
Ligand binding assays at equilibrium: validation and interpretationRadioligand Binding Assays for Determining Dissociation Constants of Phytohormone Receptors.Characterizing low affinity epibatidine binding to α4β2 nicotinic acetylcholine receptors with ligand depletion and nonspecific bindingFevipiprant (QAW039), a Slowly Dissociating CRTh2 Antagonist with the Potential for Improved Clinical Efficacy.Synthesis and characterization of [³H]-SN56, a novel radioligand for the σ₁ receptor.Long Receptor Residence Time of C26 Contributes to Super Agonist Activity at the Human β2 Adrenoceptor.Simulating the influence of plasma protein on measured receptor affinity in biochemical assays reveals the utility of Schild analysis for estimating compound affinity for plasma proteins.Extrapyramidal side effects of antipsychotics are linked to their association kinetics at dopamine D2 receptors.Reassessment of the pharmacology of Sphingosine-1-phosphate S1P3 receptor ligands using the DiscoveRx PathHunter™ and Ca2+ release functional assays.Expression, Functional Characterization, and Solid-State NMR Investigation of the G Protein-Coupled GHS Receptor in Bilayer MembranesSlow receptor dissociation is not a key factor in the duration of action of inhaled long-acting β2-adrenoceptor agonistsVersatility of homogeneous time-resolved fluorescence resonance energy transfer assays for biologics drug discovery.An Invitation to Pharmacostatics.Competition radioligand binding assays for the investigation of bispyridinium compound affinities to the human muscarinic acetylcholine receptor subtype 5 (hM(5) ).An Alternative Thiol-Reactive Dye to Analyze Ligand Interactions with the Chemokine Receptor CXCR2 Using a New Thermal Shift Assay Format.Ligand Specific Efficiency (LSE) Index for PET Tracer Optimization.Measuring receptor target coverage: a radioligand competition binding protocol for assessing the association and dissociation rates of unlabeled compounds.
P2860
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P2860
Miniaturized receptor binding assays: complications arising from ligand depletion.
description
2007 nî lūn-bûn
@nan
2007年の論文
@ja
2007年学术文章
@wuu
2007年学术文章
@zh
2007年学术文章
@zh-cn
2007年学术文章
@zh-hans
2007年学术文章
@zh-my
2007年学术文章
@zh-sg
2007年學術文章
@yue
2007年學術文章
@zh-hant
name
Miniaturized receptor binding assays: complications arising from ligand depletion.
@en
Miniaturized receptor binding assays: complications arising from ligand depletion.
@nl
type
label
Miniaturized receptor binding assays: complications arising from ligand depletion.
@en
Miniaturized receptor binding assays: complications arising from ligand depletion.
@nl
prefLabel
Miniaturized receptor binding assays: complications arising from ligand depletion.
@en
Miniaturized receptor binding assays: complications arising from ligand depletion.
@nl
P2860
P356
P1476
Miniaturized receptor binding assays: complications arising from ligand depletion.
@en
P2093
Clare M Scaramellini Carter
Juliet R Leighton-Davies
P2860
P304
P356
10.1177/1087057106297788
P577
2007-01-26T00:00:00Z