The 5-HT3B subunit confers spontaneous channel opening and altered ligand properties of the 5-HT3 receptor.
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The Concise Guide to PHARMACOLOGY 2013/14: ligand-gated ion channels.Constitutively Active 5-HT Receptors: An Explanation of How 5-HT Antagonists Inhibit Gut Motility in Species Where 5-HT is Not an Enteric Neurotransmitter?Partial agonism of 5-HT3 receptors: a novel approach to the symptomatic treatment of IBS-D5-HT3 and 5-HT4 antagonists inhibit peristaltic contractions in guinea-pig distal colon by mechanisms independent of endogenous 5-HT.The 5-HT3AB receptor shows an A3B2 stoichiometry at the plasma membrane.Direct subunit-dependent multimodal 5-hydroxytryptamine3 receptor antagonism by methadone.A single channel mutation alters agonist efficacy at 5-HT3A and 5-HT3AB receptors.Hydrophobic photolabeling studies identify the lipid-protein interface of the 5-HT3A receptor.The structural basis of function in Cys-loop receptors.The Cys-loop pentameric ligand-gated ion channel receptors: 50 years on.Cysteine modification reveals which subunits form the ligand binding site in human heteromeric 5-HT3AB receptors.Is There a Role for Endogenous 5-HT in Gastrointestinal Motility? How Recent Studies Have Changed Our Understanding.By what mechanism does ondansetron inhibit colonic migrating motor complexes: does it require endogenous serotonin in the gut wall?Structural determinants of Ca2+ permeability and conduction in the human 5-hydroxytryptamine type 3A receptor.Structure-activity relationships of quinoxaline-based 5-HT3A and 5-HT3AB receptor-selective ligands.Auto-inhibition at a ligand-gated ion channel: a cross-talk between orthosteric and allosteric sites.Agonists and antagonists induce different palonosetron dissociation rates in 5-HT₃A and 5-HT₃AB receptors.
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P2860
The 5-HT3B subunit confers spontaneous channel opening and altered ligand properties of the 5-HT3 receptor.
description
2008 nî lūn-bûn
@nan
2008 թուականի Յունուարին հրատարակուած գիտական յօդուած
@hyw
2008 թվականի հունվարին հրատարակված գիտական հոդված
@hy
2008年の論文
@ja
2008年論文
@yue
2008年論文
@zh-hant
2008年論文
@zh-hk
2008年論文
@zh-mo
2008年論文
@zh-tw
2008年论文
@wuu
name
The 5-HT3B subunit confers spo ...... perties of the 5-HT3 receptor.
@ast
The 5-HT3B subunit confers spo ...... perties of the 5-HT3 receptor.
@en
The 5-HT3B subunit confers spo ...... perties of the 5-HT3 receptor.
@nl
type
label
The 5-HT3B subunit confers spo ...... perties of the 5-HT3 receptor.
@ast
The 5-HT3B subunit confers spo ...... perties of the 5-HT3 receptor.
@en
The 5-HT3B subunit confers spo ...... perties of the 5-HT3 receptor.
@nl
prefLabel
The 5-HT3B subunit confers spo ...... perties of the 5-HT3 receptor.
@ast
The 5-HT3B subunit confers spo ...... perties of the 5-HT3 receptor.
@en
The 5-HT3B subunit confers spo ...... perties of the 5-HT3 receptor.
@nl
P2860
P356
P1476
The 5-HT3B subunit confers spo ...... perties of the 5-HT3 receptor.
@en
P2093
Robert W Peoples
Xiang-Qun Hu
P2860
P304
P356
10.1074/JBC.M707571200
P407
P577
2008-01-10T00:00:00Z