A neoceptor approach to unraveling microscopic interactions between the human A2A adenosine receptor and its agonists.
about
Adenosine receptors as therapeutic targetsEvaluation of homology modeling of G-protein-coupled receptors in light of the A(2A) adenosine receptor crystallographic structure.Structure-based approaches to ligands for G-protein-coupled adenosine and P2Y receptors, from small molecules to nanoconjugates.Recent improvements in the development of A(2B) adenosine receptor agonists.Remote control of neuronal signaling.Probing the binding site of the A1 adenosine receptor reengineered for orthogonal recognition by tailored nucleosides.Structure-activity relationships of 2,N(6),5'-substituted adenosine derivatives with potent activity at the A2B adenosine receptor.Medicinal chemistry of the A3 adenosine receptor: agonists, antagonists, and receptor engineering.Purine receptors: GPCR structure and agonist designOrthogonal activation of the reengineered A3 adenosine receptor (neoceptor) using tailored nucleoside agonists.Optimization of adenosine 5'-carboxamide derivatives as adenosine receptor agonists using structure-based ligand design and fragment screening.Probing GPCR structure: adenosine and P2Y nucleotide receptors.Action of nucleosides and nucleotides at 7 transmembrane-spanning receptors.Neoceptors: reengineering GPCRs to recognize tailored ligandsApplication of the functionalized congener approach to dendrimer-based signaling agents acting through A(2A) adenosine receptors.Novel approaches for targeting the adenosine A2A receptor.Mapping the intramolecular signal transduction of G-protein coupled receptors.Breakthrough in GPCR Crystallography and Its Impact on Computer-Aided Drug Design.Structure-Based Scaffold Repurposing for G Protein-Coupled Receptors: Transformation of Adenosine Derivatives into 5HT2B/5HT2C Serotonin Receptor Antagonists.
P2860
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P2860
A neoceptor approach to unraveling microscopic interactions between the human A2A adenosine receptor and its agonists.
description
2005 nî lūn-bûn
@nan
2005 թուականի Փետրուարին հրատարակուած գիտական յօդուած
@hyw
2005 թվականի փետրվարին հրատարակված գիտական հոդված
@hy
2005年の論文
@ja
2005年論文
@yue
2005年論文
@zh-hant
2005年論文
@zh-hk
2005年論文
@zh-mo
2005年論文
@zh-tw
2005年论文
@wuu
name
A neoceptor approach to unrave ...... ine receptor and its agonists.
@ast
A neoceptor approach to unrave ...... ine receptor and its agonists.
@en
type
label
A neoceptor approach to unrave ...... ine receptor and its agonists.
@ast
A neoceptor approach to unrave ...... ine receptor and its agonists.
@en
prefLabel
A neoceptor approach to unrave ...... ine receptor and its agonists.
@ast
A neoceptor approach to unrave ...... ine receptor and its agonists.
@en
P2093
P2860
P50
P1476
A neoceptor approach to unrave ...... ine receptor and its agonists.
@en
P2093
Heng T Duong
Michal Cesnek
Michihiro Ohno
Soo-Kyung Kim
Susanna Tchilibon
P2860
P304
P356
10.1016/J.CHEMBIOL.2004.12.010
P577
2005-02-01T00:00:00Z