A broadly applicable [18F]trifluoromethylation of aryl and heteroaryl iodides for PET imaging.
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Carbon-carbon bond cleavage for Cu-mediated aromatic trifluoromethylations and pentafluoroethylationsDecarboxylative fluorination strategies for accessing medicinally- relevant productsOne-step (18)F labeling of biomolecules using organotrifluoroboratesDevelopment and Evaluation of 18F-IRS for Molecular Imaging Mutant EGF Receptors in NSCLC.Targeted fluorination with the fluoride ion by manganese-catalyzed decarboxylation.Academia-industry symbiosis in organic chemistry.PET imaging of bacterial infections with fluorine-18-labeled maltohexaose.Boramino acid as a marker for amino acid transporters.18F-Fluoroform: a 18F-trifluoromethylating agent for the synthesis of SCF218F-aromatic derivatives.Difluorocarbene-Derived Trifluoromethylthiolation and [(18)F]Trifluoromethylthiolation of Aliphatic ElectrophilesN'-3-(Trifluoromethyl)phenyl Derivatives of N-Aryl-N'-methylguanidines as Prospective PET Radioligands for the Open Channel of the N-Methyl-d-aspartate (NMDA) Receptor: Synthesis and Structure-Affinity RelationshipsInvestigation of the Brain Biodistribution of the Lipoprotein-Associated Phospholipase A2 (Lp-PLA2) Inhibitor [18F]GSK2647544 in Healthy Male Subjects.Radiosynthesis of [18)F]trifluoroalkyl groups: scope and limitations.18F-labelled intermediates for radiosynthesis by modular build-up reactions: newer developments.Recent Advances in the One-Step Synthesis of Distally Fluorinated Ketones.Considerations in the Development of Reversibly Binding PET Radioligands for Brain Imaging.Fluorine-18 patents (2009-2015). Part 2: new radiochemistry.Synthesis of (18) F-Difluoromethylarenes from Aryl (Pseudo) HalidesAn Unconventional Mechanistic Insight into SCF3 Formation from Difluorocarbene: Preparation of 18 F-Labeled α-SCF3 Carbonyl Compounds.Photochemical Perfluoroalkylation with Pyridine N-Oxides: Mechanistic Insights and Performance on a Kilogram Scale.Late-stage [(18)F]Fluorination: New Solutions to Old ProblemsA catalytic fluoride-rebound mechanism for C(sp3)-CF3 bond formation.[11 C]Fluoroform, a Breakthrough for Versatile Labeling of PET Radiotracer Trifluoromethyl Groups in High Molar Activity.Carbon-11 radiolabelling of organosulfur compounds: (11) C synthesis of the progesterone receptor agonist tanaproget.MS565: A SPECT Tracer for Evaluating the Brain Penetration of BAF312 (Siponimod).Catalyst free synthesis of α-fluoro-β-hydroxy ketones/α-fluoro-ynols via electrophilic fluorination of tertiary propargyl alcohols using Selectfluor™ (F-TEDA-BF4).Efficient DBU accelerated synthesis of 18F-labelled trifluoroacetamides.The first nucleophilic C-H perfluoroalkylation of aromatic compounds via (arene)tricarbonylchromium complexes.Nano-graphene oxide composite for in vivo imaging.Site-Selective Tertiary Alkyl-Fluorine Bond Formation from α-Bromoamides Using a Copper/CsF Catalyst System.Highly mono-selective ortho-trifluoromethylation of benzamides via 8-aminoquinoline assisted Cu-promoted C-H activations.Silver-Mediated Oxidative Trifluoromethylation of Phenols: Direct Synthesis of Aryl Trifluoromethyl Ethers.Site-selective 18F fluorination of unactivated C-H bonds mediated by a manganese porphyrin.Radiosynthesis of the anticancer nucleoside analogue Trifluridine using an automated 18F-trifluoromethylation procedure.Mn-salen catalysed benzylic C-H activation for the synthesis of aryl [(18)F]CF3-containing PET probes.A universal procedure for the [¹⁸F]trifluoromethylation of aryl iodides and aryl boronic acids with highly improved specific activity.[(18) F]CuCF3 : a [(18) F]trifluoromethylating agent for arylboronic acids and aryl iodides.Exploiting the unusual effects of fluorine in methodology.(18)F-Labeling of Aryl-SCF3, -OCF3 and -OCHF2 with [(18)F]Fluoride.The Synthesis and Evaluation of Fluoro-, Trifluoromethyl-, and Iodomuscimols as GABA Agonists.
P2860
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P2860
A broadly applicable [18F]trifluoromethylation of aryl and heteroaryl iodides for PET imaging.
description
2013 nî lūn-bûn
@nan
2013年の論文
@ja
2013年学术文章
@wuu
2013年学术文章
@zh
2013年学术文章
@zh-cn
2013年学术文章
@zh-hans
2013年学术文章
@zh-my
2013年学术文章
@zh-sg
2013年學術文章
@yue
2013年學術文章
@zh-hant
name
A broadly applicable [18F]trif ...... oaryl iodides for PET imaging.
@en
A broadly applicable [18F]trif ...... oaryl iodides for PET imaging.
@nl
type
label
A broadly applicable [18F]trif ...... oaryl iodides for PET imaging.
@en
A broadly applicable [18F]trif ...... oaryl iodides for PET imaging.
@nl
prefLabel
A broadly applicable [18F]trif ...... oaryl iodides for PET imaging.
@en
A broadly applicable [18F]trif ...... oaryl iodides for PET imaging.
@nl
P2093
P2860
P356
P1433
P1476
A broadly applicable [18F]trif ...... oaryl iodides for PET imaging.
@en
P2093
Jan Passchier
Mickael Huiban
Satoshi Mizuta
Thomas Lee Collier
Véronique Gouverneur
Xiaomin Zhang
Zehong Wan
P2860
P2888
P304
P356
10.1038/NCHEM.1756
P577
2013-09-08T00:00:00Z