Cocrystal Structures of Primed Side-Extending α-Ketoamide Inhibitors Reveal Novel Calpain-Inhibitor Aromatic Interactions #

Cocrystal Structures of Primed Side-Extending α-Ketoamide Inhibitors Reveal Novel Calpain-Inhibitor Aromatic Interactions #

Item
http://www.wikidata.org/entity/Q27651571
Understanding the interaction determinants of CAPN1 inhibition by CAST4 from bovines using molecular modeling techniques.Peptidyl alpha-ketoamides with nucleobases, methylpiperazine, and dimethylaminoalkyl substituents as calpain inhibitorsMechanism of action of thalassospiramides, a new class of calpain inhibitorsIn silico affinity profiling of neuroactive polyphenols for post-traumatic calpain inactivation: a molecular docking and atomistic simulation sensitivity analysis.Development of α-helical calpain probes by mimicking a natural protein-protein interaction.Calpain inhibitors: a survey of compounds reported in the patent and scientific literature.Structure-function relationships in calpains.An updated patent review of calpain inhibitors (2012 - 2014).Calpain research for drug discovery: challenges and potential.Can Relative Binding Free Energy Predict Selectivity of Reversible Covalent Inhibitors?Calpain-2 as a therapeutic target for acute neuronal injury.Calpain inhibition modulates glycogen synthase kinase 3β pathways in ischemic myocardium: A proteomic and mechanistic analysis.One pot synthesis of α-ketoamides from ethylarenes and amines: a metal free difunctionalization strategy.A novel de novo CAPN5 mutation in a patient with inflammatory vitreoretinopathy, hearing loss, and developmental delay.Copper-TEMPO-catalyzed synthesis of α-ketoamides via tandem sp(3)C-H aerobic oxidation and amination of phenethyl alcohol derivatives.Cu(i)-Functionalized SBA-16: an efficient catalyst for the synthesis of α-ketoamides under moderate conditions.
P2860

Cocrystal Structures of Primed Side-Extending α-Ketoamide Inhibitors Reveal Novel Calpain-Inhibitor Aromatic Interactions #

Item
http://www.wikidata.org/entity/Q27651571
description
2008 nî lūn-bûn
@nan
2008 թուականի Սեպտեմբերին հրատարակուած գիտական յօդուած
@hyw
2008 թվականի սեպտեմբերին հրատարակված գիտական հոդված
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2008年の論文
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2008年論文
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2008年論文
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2008年論文
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2008年論文
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2008年論文
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2008年论文
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Cocrystal Structures of Primed ...... ibitor Aromatic Interactions #
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Cocrystal Structures of Primed ...... ibitor Aromatic Interactions #
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Cocrystal Structures of Primed ...... ibitor Aromatic Interactions #
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Cocrystal Structures of Primed ...... ibitor Aromatic Interactions #
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Cocrystal Structures of Primed ...... ibitor Aromatic Interactions #
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Cocrystal Structures of Primed ...... ibitor Aromatic Interactions #
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Cocrystal Structures of Primed ...... ibitor Aromatic Interactions #
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Cocrystal Structures of Primed ...... ibitor Aromatic Interactions #
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Cocrystal Structures of Primed ...... ibitor Aromatic Interactions #
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Cocrystal structures of primed ...... nhibitor aromatic interactions
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P356
P407
P433
P478
P50
P577
P5875
P698
P921
P932