Optimisation of a triazolopyridine based histone demethylase inhibitor yields a potent and selective KDM2A (FBXL11) inhibitor
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8-Substituted Pyrido[3,4-d]pyrimidin-4(3H)-one Derivatives As Potent, Cell Permeable, KDM4 (JMJD2) and KDM5 (JARID1) Histone Lysine Demethylase InhibitorsPotent and Selective KDM5 Inhibitor Stops Cellular Demethylation of H3K4me3 at Transcription Start Sites and Proliferation of MM1S Myeloma Cells.Lysine demethylase 2A promotes stemness and angiogenesis of breast cancer by upregulating Jagged1Inhibitors of Protein Methyltransferases and Demethylases.Histone Lysine Demethylase Inhibitors.Discovery of a Highly Selective Cell-Active Inhibitor of the Histone Lysine Demethylases KDM2/7.Small molecule KDM4s inhibitors as anti-cancer agents.Discovery of a Highly Selective Cell-Active Inhibitor of the Histone Lysine Demethylases KDM2/7
P2860
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P2860
Optimisation of a triazolopyridine based histone demethylase inhibitor yields a potent and selective KDM2A (FBXL11) inhibitor
description
2014 nî lūn-bûn
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2014年の論文
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2014年論文
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2014年論文
@zh-hant
2014年論文
@zh-hk
2014年論文
@zh-mo
2014年論文
@zh-tw
2014年论文
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2014年论文
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2014年论文
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name
Optimisation of a triazolopyri ...... ctive KDM2A (FBXL11) inhibitor
@ast
Optimisation of a triazolopyri ...... ctive KDM2A (FBXL11) inhibitor
@en
type
label
Optimisation of a triazolopyri ...... ctive KDM2A (FBXL11) inhibitor
@ast
Optimisation of a triazolopyri ...... ctive KDM2A (FBXL11) inhibitor
@en
prefLabel
Optimisation of a triazolopyri ...... ctive KDM2A (FBXL11) inhibitor
@ast
Optimisation of a triazolopyri ...... ctive KDM2A (FBXL11) inhibitor
@en
P2093
P2860
P50
P356
P1433
P1476
Optimisation of a triazolopyri ...... ctive KDM2A (FBXL11) inhibitor
@en
P2093
Aleksandra Szykowska
Anthony Tumber
Giuseppe Scozzafava
KaHing Che
Katherine S England
Michelle Daniel
Nicola A Burgess-Brown
Paul E Brennan
Stanley S Ng
P2860
P304
P356
10.1039/C4MD00291A
P577
2014-12-01T00:00:00Z