A systematic approach to diverse, lead-like scaffolds from α,α-disubstituted amino acids.
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Evaluating New Chemistry to Drive Molecular Discovery: Fit for Purpose?A divergent synthetic approach to diverse molecular scaffolds: assessment of lead-likeness using LLAMA, an open-access computational tool.Ring-Expansion Approach to Medium-Sized Lactams and Analysis of Their Medicinal Lead-Like Properties.Synthesis of sp(3)-rich scaffolds for molecular libraries through complexity-generating cascade reactions.A metal-catalyzed enyne-cyclization step for the synthesis of bi- and tricyclic scaffolds amenable to molecular library production.Scaffold Diversity Synthesis and Its Application in Probe and Drug Discovery.Palladium-Catalyzed Directed C(sp(3))-H Arylation of Saturated Heterocycles at C-3 Using a Concise Optimization ApproachSelective Synthesis of Six Products from a Single Indolyl α-Diazocarbonyl Precursor.Evaluierung neuer Reaktionen zur Steuerung der Wirkstoff-Forschung: ein EignungstestRecent Applications of Diversity-Oriented Synthesis Toward Novel, 3-Dimensional Fragment CollectionsRing-opening metathesis of some strained bicyclic systems; stereocontrolled access to diolefinated saturated heterocycles with multiple stereogenic centers
P2860
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P2860
A systematic approach to diverse, lead-like scaffolds from α,α-disubstituted amino acids.
description
2015 nî lūn-bûn
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2015年の論文
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2015年学术文章
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2015年学术文章
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2015年学术文章
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2015年学术文章
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2015年学术文章
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2015年学术文章
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2015年學術文章
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2015年學術文章
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name
A systematic approach to diverse, lead-like scaffolds from α,α-disubstituted amino acids.
@en
A systematic approach to diverse, lead-like scaffolds from α,α-disubstituted amino acids.
@en-gb
A systematic approach to diverse, lead-like scaffolds from α,α-disubstituted amino acids.
@nl
type
label
A systematic approach to diverse, lead-like scaffolds from α,α-disubstituted amino acids.
@en
A systematic approach to diverse, lead-like scaffolds from α,α-disubstituted amino acids.
@en-gb
A systematic approach to diverse, lead-like scaffolds from α,α-disubstituted amino acids.
@nl
prefLabel
A systematic approach to diverse, lead-like scaffolds from α,α-disubstituted amino acids.
@en
A systematic approach to diverse, lead-like scaffolds from α,α-disubstituted amino acids.
@en-gb
A systematic approach to diverse, lead-like scaffolds from α,α-disubstituted amino acids.
@nl
P2860
P50
P356
P1154
2-s2.0-84933566830
P1476
A systematic approach to diverse, lead-like scaffolds from α,α-disubstituted amino acids.
@en
P2093
Ian Churcher
P2860
P304
11174-11177
P356
10.1039/C5CC03002A
P407
P5530
P577
2015-06-01T00:00:00Z
P6179
1031568206