μ-opioid receptors: correlation of agonist efficacy for signalling with ability to activate internalization.
about
Novel GPCR paradigms at the μ-opioid receptorBiological redundancy of endogenous GPCR ligands in the gut and the potential for endogenous functional selectivityPositive allosteric modulators of the μ-opioid receptor: a novel approach for future pain medicationsOpiate agonist-induced re-distribution of Wntless, a mu-opioid receptor interacting protein, in rat striatal neuronsLigand-Based Discovery of a New Scaffold for Allosteric Modulation of the μ-Opioid Receptor.Loss of morphine reward and dependence in mice lacking G protein-coupled receptor kinase 5.Impact of efficacy at the μ-opioid receptor on antinociceptive effects of combinations of μ-opioid receptor agonists and cannabinoid receptor agonists.Identification of phosphorylation sites in the COOH-terminal tail of the μ-opioid receptorFunctionally selective signaling for morphine and fentanyl antinociception and tolerance mediated by the rat periaqueductal gray.Opioid receptor desensitization: mechanisms and its link to toleranceFunctional selectivity and time-dependence of μ-opioid receptor desensitization at nerve terminals in the mouse ventral tegmental areaChange in functional selectivity of morphine with the development of antinociceptive tolerance.Protein kinase Czeta mediates micro-opioid receptor-induced cross-desensitization of chemokine receptor CCR5.μ-Opioid receptor coupling to Gα(o) plays an important role in opioid antinociception.Quantifying ligand bias at seven-transmembrane receptors.Phosphatidylethanolamine-binding protein is not involved in µ-opioid receptor-mediated regulation of extracellular signal-regulated kinase.Agonist-directed interactions with specific beta-arrestins determine mu-opioid receptor trafficking, ubiquitination, and dephosphorylation.Functional selectivity at the μ-opioid receptor: implications for understanding opioid analgesia and tolerance.Analysis of opioid efficacy, tolerance, addiction and dependence from cell culture to humanTime course of altered sensitivity to inhibitory and excitatory agonist responses in the longitudinal muscle-myenteric plexus and analgesia in the Guinea pig after chronic morphine treatment.Tolerance to the antinociceptive effects of chronic morphine requires c-Jun N-terminal kinase.The 5-HT3B subunit affects high-potency inhibition of 5-HT3 receptors by morphineRole of G Protein-Coupled Receptor Kinases 2 and 3 in μ-Opioid Receptor Desensitization and InternalizationGRK2 protein-mediated transphosphorylation contributes to loss of function of μ-opioid receptors induced by neuropeptide FF (NPFF2) receptors.Differences in the characteristics of tolerance to μ-opioid receptor agonists in the colon from wild type and β-arrestin2 knockout miceMechanisms of rapid opioid receptor desensitization, resensitization and tolerance in brain neurons.Evidence that behavioral phenotypes of morphine in β-arr2-/- mice are due to the unmasking of JNK signaling.ßarrestin1-biased agonism at human δ-opioid receptor by peptidic and alkaloid ligands.Opioid receptors: Structural and mechanistic insights into pharmacology and signaling.Endomorphin-2: a biased agonist at the μ-opioid receptor.Ethanol Reversal of Tolerance to the Respiratory Depressant Effects of MorphineMemantine improves buprenorphine/naloxone treatment for opioid dependent young adultsModulating neuromodulation by receptor membrane traffic in the endocytic pathway.Regulation of μ-opioid receptors: desensitization, phosphorylation, internalization, and tolerance.The role of kinetic context in apparent biased agonism at GPCRs.Differentiation of opioid drug effects by hierarchical multi-site phosphorylationLigand-biased activation of extracellular signal-regulated kinase 1/2 leads to differences in opioid induced antinociception and tolerance.Propagation of conformational changes during μ-opioid receptor activation.Quantitative encoding of the effect of a partial agonist on individual opioid receptors by multisite phosphorylation and threshold detection.Reversal of morphine analgesic tolerance by ethanol in the mouse.
P2860
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P2860
μ-opioid receptors: correlation of agonist efficacy for signalling with ability to activate internalization.
description
2010 nî lūn-bûn
@nan
2010 թուականի Յուլիսին հրատարակուած գիտական յօդուած
@hyw
2010 թվականի հուլիսին հրատարակված գիտական հոդված
@hy
2010年の論文
@ja
2010年論文
@yue
2010年論文
@zh-hant
2010年論文
@zh-hk
2010年論文
@zh-mo
2010年論文
@zh-tw
2010年论文
@wuu
name
μ-opioid receptors: correlatio ...... y to activate internalization.
@ast
μ-opioid receptors: correlatio ...... y to activate internalization.
@en
μ-opioid receptors: correlatio ...... y to activate internalization.
@nl
type
label
μ-opioid receptors: correlatio ...... y to activate internalization.
@ast
μ-opioid receptors: correlatio ...... y to activate internalization.
@en
μ-opioid receptors: correlatio ...... y to activate internalization.
@nl
prefLabel
μ-opioid receptors: correlatio ...... y to activate internalization.
@ast
μ-opioid receptors: correlatio ...... y to activate internalization.
@en
μ-opioid receptors: correlatio ...... y to activate internalization.
@nl
P2093
P2860
P50
P356
P1476
μ-opioid receptors: correlatio ...... y to activate internalization.
@en
P2093
Eamonn Kelly
Graeme Henderson
Jamie McPherson
Javier Llorente
Myma Baptist
William L Dewey
P2860
P304
P356
10.1124/MOL.110.066613
P50
P577
2010-07-20T00:00:00Z