Characterization using FLIPR of rat vanilloid receptor (rVR1) pharmacology
about
Effects of piperine, the pungent component of black pepper, at the human vanilloid receptor (TRPV1)Characterization of the mouse cold-menthol receptor TRPM8 and vanilloid receptor type-1 VR1 using a fluorometric imaging plate reader (FLIPR) assayPharmacological differences between the human and rat vanilloid receptor 1 (VR1)Differential effects of anandamide on acetylcholine release in the guinea-pig ileum mediated via vanilloid and non-CB1 cannabinoid receptorsTRPA1 mediates the noxious effects of natural sesquiterpene deterrents.A pathogenic C terminus-truncated polycystin-2 mutant enhances receptor-activated Ca2+ entry via association with TRPC3 and TRPC7Activation of vanilloid receptor 1 by resiniferatoxin mobilizes calcium from inositol 1,4,5-trisphosphate-sensitive stores.Respiratory actions of vanilloid receptor agonists in the nucleus of the solitary tract: comparison of resiniferatoxin with non-pungent agents and anandamide.The effects of Delta9-tetrahydrocannabinol in rat mesenteric vasculature, and its interactions with the endocannabinoid anandamide.Increased function of the TRPV1 channel in small sensory neurons after local inflammation or in vitro exposure to the pro-inflammatory cytokine GRO/KC.A yeast genetic screen reveals a critical role for the pore helix domain in TRP channel gatingCapsaicinoids cause inflammation and epithelial cell death through activation of vanilloid receptors.Protein kinase C(alpha) is required for vanilloid receptor 1 activation. Evidence for multiple signaling pathways.Neuronal cell lines as model dorsal root ganglion neurons: A transcriptomic comparison.Thymol and related alkyl phenols activate the hTRPA1 channel.Novel gating and sensitizing mechanism of capsaicin receptor (TRPV1): tonic inhibitory regulation of extracellular sodium through the external protonation sites on TRPV1.Comparison of human recombinant adenosine A2B receptor function assessed by Fluo-3-AM fluorometry and microphysiometry.Interaction of chelerythrine with inositol phosphate metabolism.Anandamide activates vanilloid receptor 1 (VR1) at acidic pH in dorsal root ganglia neurons and cells ectopically expressing VR1.Activation of vanilloid receptor type I in the endoplasmic reticulum fails to activate store-operated Ca2+ entry.Anandamide is a partial agonist at native vanilloid receptors in acutely isolated mouse trigeminal sensory neurons.Mechanisms of acid-induced activation of airway afferent nerve fibres in guinea-pig.Use of a fluorescent imaging plate reader--based calcium assay to assess pharmacological differences between the human and rat vanilloid receptor.Identification of species-specific determinants of the action of the antagonist capsazepine and the agonist PPAHV on TRPV1.Intragastric administration of TRPV1, TRPV3, TRPM8, and TRPA1 agonists modulates autonomic thermoregulation in different manners in mice.TRPA1 agonists--allyl isothiocyanate and cinnamaldehyde--induce adrenaline secretion.Piperine, an alkaloid from black pepper, inhibits growth of human colon cancer cells via G1 arrest and apoptosis triggered by endoplasmic reticulum stress.Capsaicin-induced vasodilatation in human nasal vasculature is mediated by modulation of cyclooxygenase-2 activity and abrogated by sulprostone.Use of cryopreserved cells for enabling greater flexibility in compound profiling.
P2860
Q24670592-25B98B51-CA09-4D04-BAED-96D17239C2DDQ24672180-B7EF635A-F9DF-4401-AB60-259AD974EB47Q28115814-DB5344C7-C2E2-451B-B043-01407743CF40Q28346747-0CCC178D-D99A-4710-A274-2B31356D707BQ30483295-EDFFDF82-7030-4016-AD77-A2046956EBE9Q30492499-7A552092-BA0A-4106-A810-7AED6875FD55Q31125580-5CF93DEC-62E9-4452-8163-7FEE5FF370DAQ35044726-6F5B3A58-F5F1-4C60-8629-F1293D4E4271Q35048945-2A6C6D39-B13A-4A07-A342-147688520E50Q35882902-7CD52661-9A22-4A97-A5C6-9FCA6C49B74FQ36710217-76A0F845-A272-4324-9C19-C31BCE01DB7DQ36711779-770CFAEB-77B5-4D46-8C9B-9E7BBB27ACDAQ38287480-2F41EF8F-DDCC-4708-B5F1-3742CA70C3BBQ38447984-E7B22ACF-2166-4DDC-A4FC-B849A5CBB033Q39517524-D32235EB-8E0E-45D9-BCFA-C7A60489BC25Q40019228-1BD65030-D5F2-4686-85EA-1F44D779A3B4Q40669048-C2B10485-D053-4BDD-9118-240C123FBDB6Q42518899-223678EB-6EA7-4428-8931-E75BFFF792F0Q42829339-450AD963-4100-4318-A353-6B71B0F1B25FQ43002870-CA1EAC93-86BB-43E2-AC0A-298FBB1277BBQ43263656-9DF4B447-1002-4332-8261-6673A0CF7DBFQ44121203-973B64F3-9285-465F-96DA-7426E0633A54Q44643308-3290BEF1-590A-422C-9DC8-E6FB5C44AE68Q44762642-54FA4BD0-AC9E-4515-8E2B-48970E0853F4Q46022984-8075B027-F2B5-4425-A646-4A0CC684A57AQ46328971-DB54A8A0-E825-4801-A375-0F842A44757EQ46895149-D67B8462-CA9C-4E59-966B-4F82C3746DC4Q49064177-4BAC1B99-5FBF-49B8-8F01-546D717E5590Q51789269-F7B9AAB3-123D-49AB-8082-C85D2F85E7B6
P2860
Characterization using FLIPR of rat vanilloid receptor (rVR1) pharmacology
description
2000 nî lūn-bûn
@nan
2000 թուականի Յունիսին հրատարակուած գիտական յօդուած
@hyw
2000 թվականի հունիսին հրատարակված գիտական հոդված
@hy
2000年の論文
@ja
2000年論文
@yue
2000年論文
@zh-hant
2000年論文
@zh-hk
2000年論文
@zh-mo
2000年論文
@zh-tw
2000年论文
@wuu
name
Characterization using FLIPR of rat vanilloid receptor (rVR1) pharmacology
@ast
Characterization using FLIPR of rat vanilloid receptor (rVR1) pharmacology
@en
Characterization using FLIPR of rat vanilloid receptor (rVR1) pharmacology
@nl
type
label
Characterization using FLIPR of rat vanilloid receptor (rVR1) pharmacology
@ast
Characterization using FLIPR of rat vanilloid receptor (rVR1) pharmacology
@en
Characterization using FLIPR of rat vanilloid receptor (rVR1) pharmacology
@nl
prefLabel
Characterization using FLIPR of rat vanilloid receptor (rVR1) pharmacology
@ast
Characterization using FLIPR of rat vanilloid receptor (rVR1) pharmacology
@en
Characterization using FLIPR of rat vanilloid receptor (rVR1) pharmacology
@nl
P2093
P2860
P3181
P356
P1476
Characterization using FLIPR of rat vanilloid receptor (rVR1) pharmacology
@en
P2093
P2860
P304
P3181
P356
10.1038/SJ.BJP.0703390
P407
P577
2000-06-01T00:00:00Z