Exploration and optimization of substituted triazolothiadiazines and triazolopyridazines as PDE4 inhibitors
about
Chemical genetic screening for compounds that preferentially inhibit growth of methylthioadenosine phosphorylase (MTAP)-deficient Saccharomyces cerevisiaePhosphodiesterase 4 inhibitors enhance sexual pleasure-seeking activity in rodents.In-vivo detection of binary PKA network interactions upon activation of endogenous GPCRsSafety and efficacy of new 3,6-diaryl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine analogs as potential phosphodiesterase-4 inhibitors in NIH-3T3 mouse fibroblastic cells.
P2860
Exploration and optimization of substituted triazolothiadiazines and triazolopyridazines as PDE4 inhibitors
description
2009 nî lūn-bûn
@nan
2009 թուականի Յունուարին հրատարակուած գիտական յօդուած
@hyw
2009 թվականի հունվարին հրատարակված գիտական հոդված
@hy
2009年の論文
@ja
2009年論文
@yue
2009年論文
@zh-hant
2009年論文
@zh-hk
2009年論文
@zh-mo
2009年論文
@zh-tw
2009年论文
@wuu
name
Exploration and optimization o ...... pyridazines as PDE4 inhibitors
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Exploration and optimization o ...... pyridazines as PDE4 inhibitors
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type
label
Exploration and optimization o ...... pyridazines as PDE4 inhibitors
@ast
Exploration and optimization o ...... pyridazines as PDE4 inhibitors
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prefLabel
Exploration and optimization o ...... pyridazines as PDE4 inhibitors
@ast
Exploration and optimization o ...... pyridazines as PDE4 inhibitors
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P2093
P2860
P50
P1476
Exploration and optimization o ...... pyridazines as PDE4 inhibitors
@en
P2093
Amanda P Skoumbourdis
Christopher A Leclair
Craig J Thomas
Douglas S Auld
James Inglese
Menghang Xia
Ruili Huang
Stephen W Michnick
Steven A Titus
William Maguire
P2860
P304
P356
10.1016/J.BMCL.2009.01.057
P407
P577
2009-01-23T00:00:00Z