TIPP[psi]: a highly potent and stable pseudopeptide delta opioid receptor antagonist with extraordinary delta selectivity.
about
G-protein-coupled receptor heterodimerization modulates receptor functionStructural basis for bifunctional peptide recognition at human δ-opioid receptorThe atypical antidepressant and neurorestorative agent tianeptine is a μ-opioid receptor agonistMu and Delta opioid receptors activate the same G proteins in human neuroblastoma SH-SY5Y cellsLong-lasting antinociceptive effects of a novel dynorphin analogue, Tyr-D-Ala-Phe-Leu-Arg psi (CH(2)NH) Arg-NH(2), in miceSynaptic actions of neuropeptide FF in the rat parabrachial nucleus: interactions with opioid receptorsThe Concise Guide to PHARMACOLOGY 2013/14: G protein-coupled receptorsSubtleties of structure-agonist versus antagonist relationships of opioid peptides and peptidomimetics.The TIPP opioid peptide family: development of delta antagonists, delta agonists, and mixed mu agonist/delta antagonists.New 2',6'-dimethyl-L-tyrosine (Dmt) opioid peptidomimetics based on the Aba-Gly scaffold. Development of unique mu-opioid receptor ligandsFrog skin opioid peptides: a case for environmental mimicry.Dmt and opioid peptides: a potent alliance.Delta opioidmimetic antagonists: prototypes for designing a new generation of ultraselective opioid peptides.Molecular Pharmacology of δ-Opioid Receptors.N-terminal guanidinylation of TIPP (Tyr-Tic-Phe-Phe) peptides results in major changes of the opioid activity profile.Agonist vs antagonist behavior of delta opioid peptides containing novel phenylalanine analogues in place of Tyr(1).The role of δ-opioid receptors in learning and memory underlying the development of addiction.The design of multitarget ligands for chronic and neuropathic pain.The delta opioid receptor tool box.Characterization of opioid receptor types and subtypes with new ligands.Activation of peripheral delta opioid receptors increases cardiac tolerance to arrhythmogenic effect of ischemia/reperfusion.A chimeric opioid peptide with mixed mu agonist/delta antagonist properties.Opioid diketopiperazines: synthesis and activity of a prototypic class of opioid antagonists.Two delta opioid receptor subtypes are functional in single ventral tegmental area neurons, and can interact with the mu opioid receptor.Decreasing the configurational entropy and the hydrophobicity of EBV-derived peptide 11389 increased its antigenicity, immunogenicity and its ability of inducing IL-6.Intra-VTA deltorphin, but not DPDPE, induces place preference in ethanol-drinking rats: distinct DOR-1 and DOR-2 mechanisms control ethanol consumption and reward.
P2860
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P2860
TIPP[psi]: a highly potent and stable pseudopeptide delta opioid receptor antagonist with extraordinary delta selectivity.
description
1993 nî lūn-bûn
@nan
1993年の論文
@ja
1993年論文
@yue
1993年論文
@zh-hant
1993年論文
@zh-hk
1993年論文
@zh-mo
1993年論文
@zh-tw
1993年论文
@wuu
1993年论文
@zh
1993年论文
@zh-cn
name
TIPP[psi]: a highly potent and ...... traordinary delta selectivity.
@en
TIPP[psi]: a highly potent and ...... traordinary delta selectivity.
@nl
type
label
TIPP[psi]: a highly potent and ...... traordinary delta selectivity.
@en
TIPP[psi]: a highly potent and ...... traordinary delta selectivity.
@nl
prefLabel
TIPP[psi]: a highly potent and ...... traordinary delta selectivity.
@en
TIPP[psi]: a highly potent and ...... traordinary delta selectivity.
@nl
P2093
P356
P1476
TIPP[psi]: a highly potent and ...... traordinary delta selectivity.
@en
P2093
P304
P356
10.1021/JM00073A020
P407
P577
1993-10-01T00:00:00Z