Development of an activity-based probe and in silico design reveal highly selective inhibitors for diacylglycerol lipase-α in brain.
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Combining cross-metathesis and activity-based protein profiling: new β-lactone motifs for targeting serine hydrolasesImmunomodulatory lysophosphatidylserines are regulated by ABHD16A and ABHD12 interplay.Inhibiting endocannabinoid biosynthesis: a novel approach to the treatment of constipation.Comprehensive Analysis of Structure-Activity Relationships of α-Ketoheterocycles as sn-1-Diacylglycerol Lipase α InhibitorsRapid and profound rewiring of brain lipid signaling networks by acute diacylglycerol lipase inhibition.The novel, orally available and peripherally restricted selective cannabinoid CB2 receptor agonist LEI-101 prevents cisplatin-induced nephrotoxicity.Diacylglycerol lipase disinhibits VTA dopamine neurons during chronic nicotine exposure.Cannabinoid CB2 receptor ligand profiling reveals biased signalling and off-target activity.Highly Selective, Reversible Inhibitor Identified by Comparative Chemoproteomics Modulates Diacylglycerol Lipase Activity in Neurons.A novel live cell assay to measure diacylglycerol lipase α activityActivity-Based Probes for 15-Lipoxygenase-1.A natural substrate-based fluorescence assay for inhibitor screening on diacylglycerol lipase α.A flow cytometry assay to quantify intercellular exchange of membrane components.Liposomal Delivery of Diacylglycerol Lipase-Beta Inhibitors to Macrophages Dramatically Enhances Selectivity and Efficacy in Vivo.Bicyclic enol cyclocarbamates inhibit penicillin-binding proteins.Activity-based protein profiling reveals off-target proteins of the FAAH inhibitor BIA 10-2474.Competitive ABPP of Serine Hydrolases: A Case Study on DAGL-Alpha.Chemical Proteomic Analysis of Serine Hydrolase Activity in Niemann-Pick Type C Mouse BrainChemoproteomic Evaluation of the Polyacetylene Callyspongynic AcidDevelopment of a Multiplexed Activity-Based Protein Profiling Assay to Evaluate Activity of Endocannabinoid Hydrolase Inhibitors
P2860
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P2860
Development of an activity-based probe and in silico design reveal highly selective inhibitors for diacylglycerol lipase-α in brain.
description
2013 nî lūn-bûn
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2013年の論文
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2013年学术文章
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2013年学术文章
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2013年学术文章
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2013年学术文章
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2013年学术文章
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name
Development of an activity-bas ...... cylglycerol lipase-α in brain.
@en
Development of an activity-bas ...... cylglycerol lipase-α in brain.
@nl
type
label
Development of an activity-bas ...... cylglycerol lipase-α in brain.
@en
Development of an activity-bas ...... cylglycerol lipase-α in brain.
@nl
prefLabel
Development of an activity-bas ...... cylglycerol lipase-α in brain.
@en
Development of an activity-bas ...... cylglycerol lipase-α in brain.
@nl
P2093
P2860
P50
P356
P1476
Development of an activity-bas ...... cylglycerol lipase-α in brain.
@en
P2093
Annelot C M van Esbroeck
Gijsbert A van der Marel
Hans den Dulk
Hans van den Elst
Jaap Brouwer
Marco Allarà
Mario van der Stelt
Nico Meeuwenoord
Vincenzo Di Marzo
P2860
P304
12081-12085
P356
10.1002/ANIE.201306295
P407
P577
2013-10-31T00:00:00Z