Dynamic combinatorial chemistry employing boronic acids/boronate esters leads to potent oxygenase inhibitors.
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Protein-Directed Dynamic Combinatorial Chemistry: A Guide to Protein Ligand and Inhibitor DiscoveryOxime side-chain cross-links in an α-helical coiled-coil protein: structure, thermodynamics, and folding-templated synthesis of bicyclic speciesStructure-based design of inhibitors of the aspartic protease endothiapepsin by exploiting dynamic combinatorial chemistryFragment Linking and Optimization of Inhibitors of the Aspartic Protease Endothiapepsin: Fragment-Based Drug Design Facilitated by Dynamic Combinatorial ChemistryA strategy based on nucleotide specificity leads to a subfamily-selective and cell-active inhibitor of N6-methyladenosine demethylase FTO.Reporter ligand NMR screening method for 2-oxoglutarate oxygenase inhibitors.Dynamic combinatorial/covalent chemistry: a tool to read, generate and modulate the bioactivity of compounds and compound mixtures.Dynamic combinatorial chemistry: a tool to facilitate the identification of inhibitors for protein targets.Protein-Templated Fragment Ligations-From Molecular Recognition to Drug Discovery.Dynamic multivalency for carbohydrate-protein recognition through dynamic combinatorial libraries based on Fe(II)-bipyridine complexes.A "dial-a-receptor" dynamic combinatorial library.Dynamic combinatorial chemistry with diselenides and disulfides in water.An "ingredients" approach to functional self-synthesizing materials: a metal-ion-selective, multi-responsive, self-assembled hydrogel.An allosteric receptor by simultaneous "casting" and "molding" in a dynamic combinatorial library.Salt-induced adaptation of a dynamic combinatorial library of pseudopeptidic macrocycles: unraveling the electrostatic effects in mixed aqueous media.Reversible linkage of two distinct small molecule inhibitors of Myc generates a dimeric inhibitor with improved potency that is active in myc over-expressing cancer cell lines.Small-molecule auxin inhibitors that target YUCCA are powerful tools for studying auxin function.Affinity-Based Fluorescence Polarization Assay for High-Throughput Screening of Prolyl Hydroxylase 2 InhibitorsNMR-filtered virtual screening leads to non-metal chelating metallo-β-lactamase inhibitorsProbing secondary interactions in biomolecular recognition by dynamic combinatorial chemistry.Recent Advances in Developing Inhibitors for Hypoxia-Inducible Factor Prolyl Hydroxylases and Their Therapeutic Implications.Target-directed Dynamic Combinatorial Chemistry: A Study on Potentials and Pitfalls as Exemplified on a Bacterial Target.Sugar-boronate ester scaffold tethered pyridyl-imine palladium(II) complexes: synthesis and their in vitro anticancer evaluation.Design, preparation, and selection of DNA-encoded dynamic librariestrans-Symmetric Dynamic Covalent Systems: Connected Transamination and Transimination Reactions.Dynamic covalent organocatalysts discovered from catalytic systems through rapid deconvolution screeningDynamic Covalent Chemistry of Aldehyde Enamines: BiIII - and ScIII -Catalysis of Amine-Enamine Exchange.RNA-directed off/on switch of RNase H activity using boronic ester formation.
P2860
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P2860
Dynamic combinatorial chemistry employing boronic acids/boronate esters leads to potent oxygenase inhibitors.
description
2012 nî lūn-bûn
@nan
2012 թուականի Մայիսին հրատարակուած գիտական յօդուած
@hyw
2012 թվականի մայիսին հրատարակված գիտական հոդված
@hy
2012年の論文
@ja
2012年論文
@yue
2012年論文
@zh-hant
2012年論文
@zh-hk
2012年論文
@zh-mo
2012年論文
@zh-tw
2012年论文
@wuu
name
Dynamic combinatorial chemistr ...... o potent oxygenase inhibitors.
@ast
Dynamic combinatorial chemistr ...... o potent oxygenase inhibitors.
@en
Dynamic combinatorial chemistr ...... o potent oxygenase inhibitors.
@nl
type
label
Dynamic combinatorial chemistr ...... o potent oxygenase inhibitors.
@ast
Dynamic combinatorial chemistr ...... o potent oxygenase inhibitors.
@en
Dynamic combinatorial chemistr ...... o potent oxygenase inhibitors.
@nl
prefLabel
Dynamic combinatorial chemistr ...... o potent oxygenase inhibitors.
@ast
Dynamic combinatorial chemistr ...... o potent oxygenase inhibitors.
@en
Dynamic combinatorial chemistr ...... o potent oxygenase inhibitors.
@nl
P2093
P2860
P50
P356
P1476
Dynamic combinatorial chemistr ...... to potent oxygenase inhibitors
@en
P2093
Kar Kheng Yeoh
Marina Demetriades
Mun Chiang Chan
Timothy D W Claridge
Ya-Min Tian
P2860
P304
P356
10.1002/ANIE.201202000
P407
P50
P577
2012-05-25T00:00:00Z