Antimalarial activities of novel synthetic cysteine protease inhibitors.

Antimalarial activities of novel synthetic cysteine protease inhibitors.

Item
http://www.wikidata.org/entity/Q34231399
Potencies of human immunodeficiency virus protease inhibitors in vitro against Plasmodium falciparum and in vivo against murine malariaBlocking Plasmodium falciparum development via dual inhibition of hemoglobin degradation and the ubiquitin proteasome system by MG132Hemoglobin cleavage site-specificity of the Plasmodium falciparum cysteine proteases falcipain-2 and falcipain-3.Plasmodium falciparum cysteine protease falcipain-1 is not essential in erythrocytic stage malaria parasites.Novel anti-plasmodial hits identified by virtual screening of the ZINC database.Antimalarial drug therapy: the role of parasite biology and drug resistance.Plasmodium yoelii inhibitor of cysteine proteases is exported to exomembrane structures and interacts with yoelipain-2 during asexual blood-stage development.Falcipain inhibitors as potential therapeutics for resistant strains of malaria: a patent review.Design, Synthesis, and Biological Evaluation of Peptidomimetic N-Substituted Cbz-4-Hyp-Hpa-Amides as Novel Inhibitors of Plasmodium falciparum.2-(3,4-dihydro-4-oxothieno[2,3-d]pyrimidin-2-ylthio) acetamides as a new class of falcipain-2 inhibitors. 3. design, synthesis and biological evaluation.BDA-410: a novel synthetic calpain inhibitor active against blood stage malaria.Analysis of non-peptidic compounds as potential malarial inhibitors against Plasmodial cysteine proteases via integrated virtual screening workflow.QSAR analysis of benzophenone derivatives as antimalarial agents.2-amido-3-(1H-indol-3-yl)-N-substituted-propanamides as a new class of falcipain-2 inhibitors. 1. Design, synthesis, biological evaluation and binding model studies.Target-similarity search using Plasmodium falciparum proteome identifies approved drugs with anti-malarial activity and their possible targets.Design, synthesis and biological evaluation of potent azadipeptide nitrile inhibitors and activity-based probes as promising anti-Trypanosoma brucei agents.
P2860

Antimalarial activities of novel synthetic cysteine protease inhibitors.

Item
http://www.wikidata.org/entity/Q34231399
description
2003 nî lūn-bûn
@nan
2003 թուականի Դեկտեմբերին հրատարակուած գիտական յօդուած
@hyw
2003 թվականի դեկտեմբերին հրատարակված գիտական հոդված
@hy
2003年の論文
@ja
2003年論文
@yue
2003年論文
@zh-hant
2003年論文
@zh-hk
2003年論文
@zh-mo
2003年論文
@zh-tw
2003年论文
@wuu
name
Antimalarial activities of novel synthetic cysteine protease inhibitors.
@ast
Antimalarial activities of novel synthetic cysteine protease inhibitors.
@en
Antimalarial activities of novel synthetic cysteine protease inhibitors.
@nl
type
label
Antimalarial activities of novel synthetic cysteine protease inhibitors.
@ast
Antimalarial activities of novel synthetic cysteine protease inhibitors.
@en
Antimalarial activities of novel synthetic cysteine protease inhibitors.
@nl
prefLabel
Antimalarial activities of novel synthetic cysteine protease inhibitors.
@ast
Antimalarial activities of novel synthetic cysteine protease inhibitors.
@en
Antimalarial activities of novel synthetic cysteine protease inhibitors.
@nl
P1433
P1476
P2093
P2860
P304
P31
P356
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P433
P478
P50
P577
P5875
P698
P921
P932
P356
P1433
P1476
Antimalarial activities of novel synthetic cysteine protease inhibitors.
@en
P2093
P2860
P304
P31
P356
10.1128/AAC.47.12.3810-3814.2003
P407
P433
P478
P50
P577
P5875
P698
P921
P932