N,N-dimethyl-thioamphetamine and methyl-thioamphetamine, two non-neurotoxic substrates of 5-HT transporters, have scant in vitro efficacy for the induction of transporter-mediated 5-HT release and currents.
about
The N terminus of monoamine transporters is a lever required for the action of amphetaminesEvidence for noncompetitive modulation of substrate-induced serotonin release.Studies of the biogenic amine transporters. 14. Identification of low-efficacy "partial" substrates for the biogenic amine transportersThe reverse operation of Na(+)/Cl(-)-coupled neurotransmitter transporters--why amphetamines take two to tango.Evidence for a role of transporter-mediated currents in the depletion of brain serotonin induced by serotonin transporter substrates.'Second-generation' mephedrone analogs, 4-MEC and 4-MePPP, differentially affect monoamine transporter function.A quantitative model of amphetamine action on the 5-HT transporter.4-Methylthioamphetamine increases dopamine in the rat striatum and has rewarding effects in vivo.Improving amphetamine therapeutic selectivity: N,N-dimethyl-MTA has dopaminergic effects and does not produce aortic contraction.
P2860
Q33796294-86EBE00D-8559-42A8-AE91-36ABDA7A9476Q34135689-99E06500-C191-4E89-A897-81FA06FA0604Q34249270-CA146544-6212-4B9D-946D-5D4C93907E24Q37627941-B9DBA90B-FC5A-4183-8BB1-F64A8BEC5C2EQ37705731-0C2EC878-226A-40EF-950C-73996D2366F3Q39644366-AA612BDB-4F0E-4F7D-914A-AEA318139CEFQ41956579-169C620A-F197-47AD-83B3-AC09D6F59828Q43964442-25E2787F-8FB8-4292-BC95-21E38AC649BFQ48821854-F46B390C-42D1-4690-B630-298F41EAAB3F
P2860
N,N-dimethyl-thioamphetamine and methyl-thioamphetamine, two non-neurotoxic substrates of 5-HT transporters, have scant in vitro efficacy for the induction of transporter-mediated 5-HT release and currents.
description
2008 nî lūn-bûn
@nan
2008年の論文
@ja
2008年論文
@yue
2008年論文
@zh-hant
2008年論文
@zh-hk
2008年論文
@zh-mo
2008年論文
@zh-tw
2008年论文
@wuu
2008年论文
@zh
2008年论文
@zh-cn
name
N,N-dimethyl-thioamphetamine a ...... ted 5-HT release and currents.
@ast
N,N-dimethyl-thioamphetamine a ...... ted 5-HT release and currents.
@en
type
label
N,N-dimethyl-thioamphetamine a ...... ted 5-HT release and currents.
@ast
N,N-dimethyl-thioamphetamine a ...... ted 5-HT release and currents.
@en
prefLabel
N,N-dimethyl-thioamphetamine a ...... ted 5-HT release and currents.
@ast
N,N-dimethyl-thioamphetamine a ...... ted 5-HT release and currents.
@en
P2093
P2860
P50
P1476
N,N-dimethyl-thioamphetamine a ...... ated 5-HT release and currents
@en
P2093
Katia Gysling
Klaus Gerstbrein
Marcella Funicello
Marion Holy
María Inés Forray
Miguel Reyes-Parada
Ramón Sotomayor
Silvio Paluzzi
Tiziana Mennini
P2860
P304
P356
10.1111/J.1471-4159.2008.05272.X
P407
P577
2008-02-04T00:00:00Z