High-throughput screening of antagonists for the orphan G-protein coupled receptor GPR139
about
Discovery and pharmacological effects of a novel GPR142 antagonist.Novel Agonist Bioisosteres and Common Structure-Activity Relationships for The Orphan G Protein-Coupled Receptor GPR139.The orphan G protein-coupled receptor GPR139 is activated by the peptides: Adrenocorticotropic hormone (ACTH), α-, and β-melanocyte stimulating hormone (α-MSH, and β-MSH), and the conserved core motif HFRW.Identification and SAR of Glycine Benzamides as Potent Agonists for the GPR139 Receptor.Re-evaluation of Adrenocorticotropic Hormone and Melanocyte Stimulating Hormone Activation of GPR139 in Vitro.Systemic and Intra-Habenular Activation of the Orphan G Protein-Coupled Receptor GPR139 Decreases Compulsive-Like Alcohol Drinking and Hyperalgesia in Alcohol-Dependent Rats.
P2860
High-throughput screening of antagonists for the orphan G-protein coupled receptor GPR139
description
2015 nî lūn-bûn
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2015年の論文
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2015年学术文章
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2015年学术文章
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2015年学术文章
@zh-hans
2015年学术文章
@zh-my
2015年学术文章
@zh-sg
2015年學術文章
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2015年學術文章
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2015年學術文章
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name
High-throughput screening of antagonists for the orphan G-protein coupled receptor GPR139
@ast
High-throughput screening of antagonists for the orphan G-protein coupled receptor GPR139
@en
type
label
High-throughput screening of antagonists for the orphan G-protein coupled receptor GPR139
@ast
High-throughput screening of antagonists for the orphan G-protein coupled receptor GPR139
@en
prefLabel
High-throughput screening of antagonists for the orphan G-protein coupled receptor GPR139
@ast
High-throughput screening of antagonists for the orphan G-protein coupled receptor GPR139
@en
P2093
P2860
P356
P1476
High-throughput screening of antagonists for the orphan G-protein coupled receptor GPR139
@en
P2093
Garrick Paul Smith
Lin-yun Zhu
Ming-wei Wang
Morten Hentzer
P2860
P2888
P304
P356
10.1038/APS.2015.12
P50
P577
2015-06-01T00:00:00Z
P5875
P6179
1032883044