Bradykinin-induced internalization of the human B2 receptor requires phosphorylation of three serine and two threonine residues at its carboxyl tail.
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Determination of bradykinin B2 receptor in vivo phosphorylation sites and their role in receptor functionAbsence of ligand-induced regulation of kinin receptor expression in the rabbitAgonist-promoted trafficking of human bradykinin receptors: arrestin- and dynamin-independent sequestration of the B2 receptor and bradykinin in HEK293 cells.The human B1 bradykinin receptor exhibits high ligand-independent, constitutive activity. Roles of residues in the fourth intracellular and third transmembrane domains.Purine and pyrimidine nucleotide-sensitive phospholipase A(2) in ampulla from frog semicircular canal.Downregulation of kinin B1 receptor function by B2 receptor heterodimerization and signaling.Kinin-stimulated B1 receptor signaling depends on receptor endocytosis whereas B2 receptor signaling does not.Mechanisms regulating the expression, self-maintenance, and signaling-function of the bradykinin B2 and B1 receptors.Structure and signalling pathways of kinin receptors.Calcium-activated potassium channels mediated blood-brain tumor barrier opening in a rat metastatic brain tumor model.Modulation of brain tumor capillaries for enhanced drug delivery selectively to brain tumor.Characterization of dual agonists for kinin B1 and B2 receptors and their biased activation of B2 receptorsAntagonist, partial agonist and antiproliferative actions of B-9870 (CU201) as a function of the expression and density of the bradykinin B1 and B2 receptorsThe G protein-coupled receptors: pharmacogenetics and disease.Conditioning the heart induces formation of signalosomes that interact with mitochondria to open mitoKATP channelsThe kallikrein-kinin system in health and in diseases of the kidney.PDE5 inhibitors enhance tumor permeability and efficacy of chemotherapy in a rat brain tumor model.Identification of functional bradykinin B(2) receptors endogenously expressed in HEK293 cells.Cardioprotective signaling to mitochondriaIcatibant , the bradykinin B2 receptor antagonist with target to the interconnected kinin systems.Targeting the 'Janus face' of the B2-bradykinin receptor.MiRNA-200b Regulates RMP7-Induced Increases in Blood-Tumor Barrier Permeability by Targeting RhoA and ROCKII.G protein-coupled receptor-mediated mitogen-activated protein kinase activation through cooperation of Galpha(q) and Galpha(i) signals.Effects of inactivation-resistant agonists on the signalling, desensitization and down-regulation of bradykinin B(2) receptors.Unraveling G protein-coupled receptor endocytosis pathways using real-time monitoring of agonist-promoted interaction between beta-arrestins and AP-2.Macrophage colony-stimulating factor differentially regulates low density lipoprotein and transferrin receptors.Expression levels strongly affect ligand-induced sequestration of B2 bradykinin receptors in transfected cells.Structural insight into the role of the second intracellular loop of the bradykinin 2 receptor in signaling and internalization.Role of hydroxyl containing residues in the intracellular region of rat bradykinin B(2) receptor in signal transduction, receptor internalization, and resensitization.Wortmannin alters the intracellular trafficking of the bradykinin B2 receptor: role of phosphoinositide 3-kinase and Rab5.Bradykinin increases intracellular calcium levels in rat testis peritubular cells via the B2 receptor subtype.Ligand-mediated regulation of kinin receptors in the rabbit.Interactions of histamine and bradykinin on polymodal C-fibres in isolated rat skin.Mechanisms underlying the contraction induced by bradykinin in the guinea pig epithelium-denuded trachea.Effects of N-, P/Q- and L-type calcium channel blockers on nociceptive neurones of the trigeminal nucleus with input from the dura.
P2860
Q28214160-11F28F6E-0F35-4ACB-A9D6-C205328DE499Q28345492-C799FE0A-FFE6-4C97-9236-39C9B3C3964FQ30664242-B7737200-0E06-438A-A842-B2BFAC38D8E8Q31778105-02D138F2-D7BF-45D6-A83B-B173F34B2F41Q32031733-6C67DA24-0D7A-4D55-8054-C176D82AD80AQ34617439-DAA8E24C-7E63-4149-97ED-A0B85A8A2E7AQ34915658-47D2EB2C-88FA-4DC4-8FDA-090B734EEFF3Q34972782-F15A775C-82D1-4C91-946C-DF25830BBF80Q35056755-99AABCE1-BDF0-487E-A253-22D7ABD60C1EQ35695284-1C11F1BE-048A-44EC-B02B-CED3E80406DFQ35778571-AEB72550-358D-40F7-90E4-11F47DB053AEQ35996074-290D695A-7155-4C9A-8F1C-104A3CAFAFE6Q36052584-69D7931E-B832-40A5-87F8-4A3D0C09B61CQ36310854-87EA38FF-E533-4E76-A232-F68070FD5B73Q36893383-7113D4C0-FA12-4B29-BC3C-D6FA35B033C8Q37070150-D5A73BFD-74EE-4AC3-A93A-3EB924A63DC1Q37076589-9702E1E6-D80E-4B9A-9215-9F9C7C3BD875Q37102919-386AE4F0-FB82-406F-81DC-1D9E1509929FQ37360936-51263BF8-743B-4010-8AFA-21AF30E1305AQ38042696-7414706D-1236-46C2-9E4E-F27C88BEDD8EQ38129928-B412CB8E-96F9-4807-A6E7-EA55A608EB4FQ38264654-46400B6D-5A91-4F6A-800A-97F4763FCF6EQ39455475-39D15696-73EE-4693-99F4-73B29DB1DC1FQ39794304-0F1500C7-4C81-400F-BA7E-587D807E4A77Q40098301-CDFB5E73-0988-49B8-AC7C-E597E7B59023Q40542671-ED095044-8EFF-48AA-9A7C-344278F85D8CQ40648440-F575A14E-0CF4-4990-B04D-EAB807F34A9DQ40755355-67E03762-85F1-4426-92F4-3A663D15B995Q40775414-68E43994-5CF9-46E0-B0C2-D8B9F7DD89C0Q41768054-9964184C-C1A0-4C1B-BDA0-EDEC446E2E1AQ43263544-A0BAC34A-668A-43D6-B298-36E02FD71021Q43547447-7490C4DE-25C3-44C2-A9C2-0CAC0061A65FQ43631748-E2F4C1E3-26D9-41B7-AC3B-12280157EC58Q44003411-DADC88E1-9179-4E4E-A11C-1A700961A234Q47927136-08B1C89A-51B3-4426-8967-2A57AC7AA725
P2860
Bradykinin-induced internalization of the human B2 receptor requires phosphorylation of three serine and two threonine residues at its carboxyl tail.
description
1999 nî lūn-bûn
@nan
1999年の論文
@ja
1999年学术文章
@wuu
1999年学术文章
@zh-cn
1999年学术文章
@zh-hans
1999年学术文章
@zh-my
1999年学术文章
@zh-sg
1999年學術文章
@yue
1999年學術文章
@zh
1999年學術文章
@zh-hant
name
Bradykinin-induced internaliza ...... residues at its carboxyl tail.
@en
type
label
Bradykinin-induced internaliza ...... residues at its carboxyl tail.
@en
prefLabel
Bradykinin-induced internaliza ...... residues at its carboxyl tail.
@en
P2093
P2860
P356
P1476
Bradykinin-induced internaliza ...... residues at its carboxyl tail
@en
P2093
F Alhenc-Gelas
R M Rajerison
P2860
P304
12738-12747
P356
10.1074/JBC.274.18.12738
P407
P577
1999-04-01T00:00:00Z